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2-[9-(5-methylthiophene-2-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
3-chloro-4-fluoro-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-benzothiophene-2-carboxamide
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
1'-(2,1,3-benzoxadiazol-4-ylmethyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(3R,4S)-4-cyclopropyl-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl]-2-methanesulfonamidoacetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4-difluorobenzamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-[2-(pyridin-3-yl)ethyl]benzamide
1-[3-(2,4-dimethoxyphenyl)propyl]-1H-imidazole
(3R,5S)-N-butyl-5-[(4-methylpiperazin-1-yl)methyl]-1-(2-phenylethyl)piperidine-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylpropanamide
3-(3-fluorophenyl)-4-(oxane-4-carbonyl)piperazin-2-one
1-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
5-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
N-[2-(2-methoxyphenyl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
3-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-[1-(2,5-dimethylphenyl)-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
2-(5-acetylthiophen-3-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
2-(dimethylamino)-N-(5-hydroxy-4,4-dimethylpentyl)-2-(2-methylphenyl)acetamide
N,N-dimethyl-3-[4-(methylsulfanyl)benzoyl]piperidine-1-sulfonamide
N-(2-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
4-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1,4-oxazepane
1-(4-benzylpiperazin-1-yl)-3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
3-(2-methylpiperidin-1-yl)-N-[2-(morpholin-4-ylmethyl)phenyl]azetidine-1-carboxamide
N-[(2R,3R)-2-methoxy-1'-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
N-(1-methoxybutan-2-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1-methyl-3-phenyl-8-[2-(propan-2-ylsulfanyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
3-[1-(2-acetylbenzoyl)piperidin-3-yl]-N-(3-chloro-4-methoxyphenyl)propanamide
4,4-difluoro-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
1-(2,3-dihydro-1H-inden-5-yl)-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazole
3-{2-[(3R)-3-hydroxypyrrolidin-1-yl]-2-oxoethyl}-2-methyl-1-(3-phenylpropyl)-4,5,6,7-tetrahydro-1H-indol-4-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2,5-dimethylphenyl)ethan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}pyridine-4-carboxamide
1-(3-fluoropyridin-4-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3-(2-phenylethyl)piperidin-3-yl]methanol
N-(2-acetylphenyl)-4-[4-(morpholin-4-yl)piperidin-1-yl]-4-oxobutanamide
5-[(2-chlorophenyl)methyl]-5-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
2-cyclopropyl-4-hydroxy-N-[2-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
4-(2-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}ethyl)phenol
1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N4-methyl-6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-2,4-diamine
2-[4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propanoic acid
N-[(2-phenoxypyridin-3-yl)methyl]isoquinoline-5-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(2-methylphenyl)methyl]piperidine-4-carboxylic acid
3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-(1-methyl-1H-indazol-6-yl)piperidine-1-carboxamide
5-{1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}-2-(2-methylphenyl)pyrimidine
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidin-2-amine