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N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3-sulfamoylthiophene-2-carboxamide
4-[(3-propylmorpholin-4-yl)methyl]-N-(trimethyl-1H-pyrazol-4-yl)benzamide
4-methyl-2-[1-(1,2-oxazole-3-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
5-(2-cyclohexylethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
N-(4-methoxyphenyl)-3-[3-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
2-[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]acetamide
3-{2-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]ethyl}phenol
N-[2-(2-fluorophenyl)-1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]-N-methyl-3-(methylsulfanyl)propanamide
4-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}butan-1-ol
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(piperidin-1-yl)ethan-1-one
[1-(5,6-dimethylpyrazin-2-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
3-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}amino)-N-(1,3-thiazol-2-yl)propanamide
2-({[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]oxy}methyl)pyridine
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(2-oxoazepan-1-yl)propanamide
5-(4-fluorophenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-{1-tert-butyl-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-3-yl}benzamide
3-[2-(dimethylamino)ethyl]-1-[4-(furan-2-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
5-(2,6-difluorophenoxymethyl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
5-methoxy-2,4-dimethyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]benzene-1-sulfonamide
3-{2-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-(4-fluoro-2-methylbenzoyl)-1-(2-methylphenyl)piperazin-2-one
7-fluoro-2-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}quinoline-4-carboxamide
5-chloro-2-methyl-6-(quinolin-8-yl)pyrimidin-4-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(piperazin-1-yl)pyridine-3-carboxamide
1-(cyclohexylmethyl)-2-(methoxymethyl)-6-methyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
1-[2-(3-fluorophenyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
2-(cyclopropylamino)-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]acetamide
6-{4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
N-cyclohexyl-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(2-methylphenyl)methyl]acetamide
5-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
5-(propan-2-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-ethyl-2-{4-[(4-hydroxy-2,6-dimethylphenyl)methyl]piperazin-1-yl}acetamide
N-(dimethyl-1,2-oxazol-4-yl)-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-[3-(cyclohexyloxy)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}propanamide
2-phenyl-1-{4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpiperazine-1-carboxamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
(cyclobutylmethyl)({[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
5-(2-fluorophenyl)-N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1,2,4-triazin-3-amine
1-[4-(butan-2-yl)phenyl]-3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
2-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-(1H-imidazol-1-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-(4-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
3-[1-(methoxymethyl)cyclopentyl]-1-(2-methoxyphenyl)urea
[3-(2-phenylethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl]methanol
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(1H-indol-1-yl)propan-2-yl]propanamide