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8-{[(4-methylphenyl)methyl]carbamoyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-(3-phenoxypropanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{3-[(2,4-difluorophenyl)methyl]-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methanol
2-[(3,4-dimethoxyphenyl)methyl]-6-(2-methylpyrrolidine-1-carbonyl)-1,3-benzoxazole
(1S,5R)-6-[(1-ethyl-1H-indol-5-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
({5-[1-(cyclohexylmethyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(4-methyl-1H-imidazol-5-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
ethyl 1-(5-methyl-1H-pyrazole-3-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
(1R,3S)-3-(2-aminoethoxy)-7-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-7-azaspiro[3.5]nonan-1-ol
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
3-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
6,7-dimethoxy-2-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
6-[(4-hydroxypiperidin-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
(8R,9aS)-2-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-N-(4-ethoxyphenyl)-3-oxopropanamide
N,N-dimethyl-2-{[3-(pyridin-4-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-chloro-2-methyl-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]benzene-1-sulfonamide
N-[(2R,3R)-1'-(4-methoxybenzoyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-(benzyloxy)-1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
4-(azepan-1-ylmethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
N-(7-{4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl}-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl)-2-methoxyacetamide
2-(3-chlorophenyl)-N-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
1-[6-(8-methoxy-2-methylquinolin-5-yl)pyridin-2-yl]ethan-1-ol
N-(2H-1,3-benzodioxol-4-ylmethyl)-N,2,2,6,6-pentamethylpiperidin-4-amine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
2-ethyl-4-methyl-N-[2-(3-methylthiophen-2-yl)ethyl]-1,3-oxazole-5-carboxamide
3-[1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]pyridine
(benzylsulfamoyl)({2-[(2-methylquinolin-8-yl)oxy]ethyl})amine
methyl 3-(4-{[3-(2-methylphenyl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
3-{3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]pyridin-2-yl}-N,N-dimethylaniline
N-[2-(4-fluorophenyl)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}propanamide
2-(1-methyl-1H-pyrazol-3-yl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
1-[5-(dimethylamino)-2-methylphenyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
ethyl 4-{[3-(3-chlorophenyl)phenyl]carbamoyl}piperazine-1-carboxylate
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
5-[(2-methoxyethyl)(methyl)amino]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
(3S,4S)-3-hydroxy-4-[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]-1λ6-thiolane-1,1-dione
8-acetyl-2-[(5-fluoro-2-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-oxo-8-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-phenoxyazetidine
1-[1-(1-methyl-1H-indole-3-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
1-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2,2-dimethyloxane-4-carboxamide