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4-methyl-5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-thiazol-2-amine
2-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}-3-methylpyrazine
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclohexanecarboxamide
3-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-1-(4-methoxy-2-methylphenyl)urea
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
(1S,5R)-3-(1,5-dimethyl-1H-pyrrole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-ethyl-N-(4-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-benzyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}benzoic acid
methyl 2-(4-{[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]amino}phenoxy)acetate
N-[3-(3-methylphenyl)phenyl]-1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidine-3-carboxamide
5-(azocane-1-carbonyl)-1-(pyridin-2-ylmethyl)piperidin-2-one
3-{4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}propan-1-ol
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidin-3-yl]methanol
N-(4-methylphenyl)-4-(thiophene-2-sulfonyl)morpholine-2-carboxamide
N-[(4-fluorophenyl)methyl]-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
6-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,6-dimethylpyridine-3-carboxamide
(2R,6R)-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-(2-methoxyethyl)-3-{[1-(oxan-4-yl)piperidin-4-yl]oxy}benzamide
(3R,4R)-1-(6-aminopyrimidin-4-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}propan-1-one
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[3-(1H-imidazol-5-yl)phenyl]urea
2-(3-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl)ethan-1-amine
(3S)-3-ethyl-4-{2-[(2-phenylethyl)sulfanyl]pyridine-3-carbonyl}morpholine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-hydroxy-4-methylpentanamide
1-(5-{3-[1-(2-hydroxypropyl)-1H-pyrazol-3-yl]phenyl}thiophen-2-yl)ethan-1-one
N-[(4-fluorophenyl)methyl]-3-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}propanamide
N-cyclohexyl-6-fluoro-N-methyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
1-(2,5-dimethylfuran-3-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][2-methyl-1-(morpholin-4-yl)propan-2-yl]amine
N-methyl-6-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,6-dihydropyridine-3-carboxamide
4-(pyridin-3-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrimidin-2-amine
(2E)-N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-3-(3-fluorophenyl)prop-2-enamide
2-(5-chlorothiophen-2-yl)-5-ethylpyrimidine
(3aS,6aR)-5-(4,6-dimethylpyrimidin-2-yl)-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(4-{4-phenyl-1-[2-(pyridin-3-yl)ethyl]-1H-imidazol-5-yl}phenoxy)ethan-1-ol
4-{3-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
N-benzyl-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
(3S,5R)-1-(pyridin-3-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methanol
N-{4-[(trifluoromethyl)sulfanyl]phenyl}-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
N,N-dimethyl-2-{[(6-methylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)propyl]-3-(2-methylphenyl)pyrrolidin-3-ol
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-4-(pyrrolidin-3-yl)benzamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
1-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)pyrrolidin-2-one
3-(2-methylphenyl)-5-[2-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazole