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N-[1-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
5-{3-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-ethylpyrrolidin-2-one
2-(morpholin-4-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
4-[(5-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
N,2,4-trimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,3-thiazole-5-carboxamide
4-(benzyloxy)-1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
4-{5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-3-yl}pyridine
N-benzyl-5-{2,7-diazaspiro[4.5]decan-7-ylmethyl}pyrimidin-2-amine
4-(3,4-difluorobenzenesulfonyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(piperidin-1-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-(furan-2-ylmethyl)-2-methyl-N-(3-methylbutan-2-yl)-4-phenylpyrimidine-5-carboxamide
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-3-methylbut-2-en-1-one
1-(4-chlorophenyl)-N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}cyclopropane-1-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-ethyl-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
3,3-dimethyl-1-[(3-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-(2-methoxyethyl)-5-(6-oxo-1,6-dihydropyridin-3-yl)furan-2-carboxamide
N-({1-[2-(1H-imidazol-1-yl)acetyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
5-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[(3R,4S)-1-(3-hydroxypropyl)-4-propylpyrrolidin-3-yl]pyridazine-3-carboxamide
3-(4-fluorophenyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine
N-{1-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylfuran-2-carboxamide
6-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
1-(dimethylamino)-2-{4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
2,2-diethyl-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]morpholine
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrrole-2-carboxamide
(3R,5S)-1-benzyl-N-[2-(1H-indol-3-yl)ethyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
N-[2-(benzyloxy)ethyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-N5-[(6-methylpyridin-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
7-[(2,3-difluorophenyl)methyl]-2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
(1-{1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}piperidin-3-yl)methanol
ethyl 1-[(4-chloro-2-methylphenyl)carbamoyl]-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
2-methoxy-N-{1-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[4-(furan-2-yl)phenyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine-3-carboxamide
2-amino-8-hydroxy-4-(2-methoxypyrimidin-5-yl)-5H,6H-benzo[h]quinoline-3-carbonitrile
5-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
(2E)-N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-3-(4-methoxyphenyl)prop-2-enamide
(furan-2-ylmethyl)({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})(thiophen-3-ylmethyl)amine
N,N,4-trimethyl-3-({[3-(propan-2-yloxy)propyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(2R,3R,6R)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-(2-methoxyethyl)-2-(5-methyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(4-cyanophenyl)-3-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carboxamide
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}quinoline-5-carboxamide
1-(6-methylhept-5-en-2-yl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-{5-[2-(methylsulfanyl)-1,3-thiazol-4-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-[(2-fluorophenyl)methyl]-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[2-(dimethyl-1,2-oxazol-4-yl)acetamido]methyl}benzoate
2-[(dimethylamino)methyl]-N-methyl-N-(quinolin-3-ylmethyl)-1,3-thiazole-4-carboxamide