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N-(5-chloro-2-methoxyphenyl)-3-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-3-yl}propanamide
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxypyridine-4-carbonyl)-4-(2-phenoxyethyl)piperazine
(1S,5R)-3-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(pyridin-4-ylmethyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-ol
1-[3-fluoro-5-(trifluoromethyl)phenyl]-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
2-[4-(isoquinolin-5-ylmethyl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-N-methylpyridin-2-amine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[(1-methylpiperidin-4-yl)methyl]-3-(2-oxopyrrolidin-1-yl)-N-(2-phenylethyl)propanamide
1-(4-{[(1R,2S)-2-phenylcyclopropyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole
1-(benzenesulfonyl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]piperidin-4-amine
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2,5-difluorobenzamide
N-cyclopropyl-3-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl}propanamide
2-(butan-2-ylsulfanyl)-5-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)pyrimidine
3-(but-2-yn-1-yl)-5-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-({7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
4-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]-3,4-dihydro-2H-1,4-benzoxazine
5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-2-(pyridin-2-yl)pyrimidine
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[3-(methylsulfanyl)phenyl]methyl}amine
4-[(3,5-dimethoxyphenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-[3-(3-methylphenyl)phenyl]piperidin-4-amine
methyl (2S)-4-methyl-2-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)formamido]pentanoate
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
4-[5-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
2-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-2,8-diazaspiro[4.5]decane
N-(3-methylphenyl)-3-(1-{spiro[2.5]octane-1-carbonyl}piperidin-4-yl)propanamide
2-(dimethylamino)-7-(4-propylbenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-chlorophenyl)-5-(oxolan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-methyl-8-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-(3-fluorophenyl)-N-[2-(1H-imidazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}acetamide
N-(2-methylprop-2-en-1-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3-(thiophen-2-yl)propanamide
2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(4-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenyl)acetamide
2-{[2-(oxan-2-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(5-phenoxyfuran-2-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(2-hydroxyethyl)-8-[(2-methylnaphthalen-1-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(6-methylpyridine-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[5-(2-benzyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidine