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3-chloro-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyridine-4-carboxamide
methyl 4-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutanoate
3-methoxy-2,2-dimethyl-N-{1-[(3-methylphenyl)methyl]cyclopropyl}propanamide
N-methyl-5-[2-(phenylamino)pyrimidine-5-carbonyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[4-(4-{[2-(morpholin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1,4-diazepan-5-one
methyl 1-(2-methoxyethoxy)-2-oxo-8-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(3-methylphenyl)methyl]piperidin-4-yl}oxy)benzamide
2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-[4-methyl-6-(methylamino)pyrimidin-2-yl]-7-azaspiro[3.5]nonan-1-ol
7-[(3-methylphenyl)methyl]-2-[2-(pyridin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[(3S)-piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
5-(4-fluorophenyl)-4-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-2-methylpyrimidine
N2,N4-bis(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-{[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]benzamide
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
3-hydroxy-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]pyridine-2-carboxamide
2-methyl-4-[5-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)thiophen-2-yl]but-3-yn-2-ol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(pyridin-4-yloxy)piperidin-1-yl]ethan-1-one
11-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-(2,1,3-benzothiadiazol-4-yl)-1H-1,3-benzodiazole-6-carboxylic acid
2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]acetamide
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-6-ethoxyquinoline
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-[(2,4,6-trimethylphenyl)methyl]-1H-pyrazole-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-tert-butylacetamide
3,5-dimethyl-1-{1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]azetidin-3-yl}-1H-pyrazole
(4aS,8aR)-6-[(2-aminopyridin-3-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-1-[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
5-benzyl-5-(1-ethylpiperidin-4-yl)imidazolidine-2,4-dione
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-3-methoxypropan-2-ol
5-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
6-[(3-fluorophenyl)methoxy]-4-(5-oxopyrrolidine-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
[(3aS,6aS)-2-(2,6,8-trimethylquinoline-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
1-(2-cyclohexylethyl)-3-hydroxy-3-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}piperidin-2-one
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-2-(4-fluorophenyl)ethyl}-2-methoxy-N-methylacetamide
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-methyl-1-(1,2,3,4-tetrahydronaphthalen-1-yl)urea
5-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2H-1,3-benzodioxol-5-yl)-5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-1H-1,2,4-triazole
1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)diethylamine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(oxolan-2-ylmethoxy)acetamide
(5-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-4-(pyridin-3-ylmethyl)piperazine