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6-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]pyridine-2-carbonitrile
7-[(2,3-difluorophenyl)methyl]-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-[3-(2,5-difluorobenzoyl)piperidine-1-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
8-[2-(2-methoxyphenoxy)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[(cyclopropylmethyl)sulfanyl]-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
7,8-dimethyl-2-(pyrimidin-5-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]quinoline-4-carboxamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-{4-[(dimethylsulfamoyl)amino]phenyl}piperidin-4-amine
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
8-chloro-2-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}quinoline
8-[(2-hydroxy-3-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}propanamide
2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-6-fluoro-1H-1,3-benzodiazole
1-cyclohexyl-4-({4-[(3-methoxypropyl)amino]-6-methylquinazolin-2-yl}methyl)piperazin-2-one
1-(2-chlorophenyl)-3-(1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-5-(4-methoxyphenyl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-methylacetamide
N,N-diethyl-1-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
9-[(2,3-dichlorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]benzenesulfonyl}piperazine
(1S,5R)-6-(4-tert-butylbenzoyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropane-1-carboxamide
{1-[(5-ethylfuran-2-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
(3S,4R)-4-(pyridin-4-yl)-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]pyrrolidine-3-carboxylic acid
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3R,4R)-3-hydroxy-4-(morpholin-4-yl)piperidin-1-yl]propan-1-one
2-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(thiophen-3-yl)acetamide
3-[(3,4-dimethoxyphenyl)methyl]-1-methyl-5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1H-1,2,4-triazole
3-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
4-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
3-phenyl-5-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1,2,4-oxadiazole
(2R)-2-amino-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-(azocan-1-ylmethyl)-4-(6-methoxypyridin-2-yl)phenol
(3S,4R)-1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
4-oxo-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,6-dimethylquinoline-3-carboxamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclobutanecarboxamide
ethyl 5-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridine-3-carboxylate
1-{3,9-diazaspiro[5.5]undecan-3-yl}-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
(3S,4S)-3-[2-(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)-1H-imidazol-1-yl]-4-hydroxy-1λ6-thiolane-1,1-dione
N-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
methyl 4-({4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxyphenyl}formamido)butanoate
9-(2-amino-6-methoxypyrimidin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-cyclopentylphenyl)-N,N-dimethylpyridine-3-carboxamide
2-ethyl-9-[(3-methylpyridin-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{[2-(adamantan-1-yl)ethyl](methyl)amino}-1-[(2,4-difluorophenyl)methyl]azepan-2-one
2-{1-[(2S)-oxolane-2-carbonyl]azetidin-3-yl}pyridine