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{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
5-(1-{2-[(2,4,6-trimethylphenyl)carbamoyl]ethyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-[(2R,3R)-1'-(4-methylbenzoyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-methoxy-1-[1'-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-cyclopropyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,3-diol
5-fluoro-N4,N4-dimethyl-N2-(thiophen-2-ylmethyl)pyrimidine-2,4-diamine
4-(1-{1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N-[(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
1-(4-methylpiperazine-1-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-(butan-2-yl)-2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}-N-(quinolin-2-ylmethyl)acetamide
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyphenyl)piperazine
3-phenyl-N-{1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
3-[(4aR,7aS)-4-(1-ethyl-1H-pyrazole-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-{[5-(quinolin-6-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-cyclopropyl-2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetamide
(2S,4S)-N,N-diethyl-1-(3-fluorobenzoyl)-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
(3R,4R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
3-(3-chlorophenyl)-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
4-cyclobutaneamido-N-[(1R)-2-hydroxy-1-phenylethyl]benzamide
N-(furan-2-ylmethyl)-5-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1'-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}spiro[indene-1,4'-piperidine]
3-{[4-(dimethylamino)phenyl]methyl}-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-({2-[2-hydroxy-3-(4-hydroxypiperidin-1-yl)propoxy]-5-methoxyphenyl}methyl)piperidin-4-ol
methyl 3-(furan-2-amido)-6-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
1-[2-(3-methoxyphenyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-methyl-5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]phenol
2-[2-chloro-4-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)phenoxy]acetamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)adamantan-1-amine
(3S,7S)-5-[2-(methylamino)pyrimidine-5-carbonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
6-(azepan-1-yl)-N-[(3-methyloxetan-3-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
methyl 1-{3-[(4-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2,3-trimethylquinoxaline-6-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(6-fluoroquinolin-2-yl)methyl](oxolan-2-ylmethyl)amine
5-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
1-(1-benzofuran-5-ylmethyl)-3-(2-methoxyphenoxy)azetidine
1-[(5-oxopyrrolidin-2-yl)methyl]-5,5-diphenylpiperidin-2-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[2-(phenylsulfanyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{5-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-2-methylpyridine
3-ethyl-1-({1-[(4-oxo-4H-chromen-3-yl)methyl]piperidin-3-yl}methyl)urea
3-{[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}-N-(2-fluoroethyl)benzamide
2-[3-cyclopropyl-5-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
2-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-4,6-dimethylpyridine-3-carbonitrile
1-(3-chloro-4-fluorophenyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-hydroxyethyl)acetamide
3-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea