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N'-(2-tert-butylphenyl)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]butanediamide
2-cyclopentyl-9-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-({[2-(4-methoxyphenyl)phenyl]carbamoyl}amino)-N-methylpentanamide
4-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]pyridine
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3S,4R)-1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2,5-dimethylphenyl)ethan-1-one
8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
3-[1-(2,2,2-trifluoroethyl)-1H-imidazol-2-yl]phenol
7,7-dimethyl-2-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)pyridazine-4-carboxamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(1-hydroxybutan-2-yl)-3-[(2-methylprop-2-en-1-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
3-(4-fluorophenyl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-(methoxymethyl)benzamide
2-(dimethylamino)-4-oxo-N-propyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
1-benzyl-3-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-(1-{7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[3-(methylsulfanyl)propyl]-1H-1,3-benzodiazole-5-carboxamide
1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-(2-chlorophenyl)-3-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-{2-[methyl(phenyl)amino]propyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
N-(furan-2-ylmethyl)-3-[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanamide
3-methyl-1-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]butan-1-one
2-hydroxy-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
4-methyl-2-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)phenol
5-[6-methyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-(2-methoxyphenyl)-4-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}piperazine
5-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[2-(2-cyclohexylpyrimidin-5-yl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide
8-chloro-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}quinoline
2-(pyridin-2-ylmethyl)-8-(quinolin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-1-(2-aminopyrimidin-4-yl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-ethyl-N-[(1R,2S)-2-phenylcyclohexyl]-1H-pyrazole-5-carboxamide
1-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]-4-phenylpiperazine
ethyl 5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
3-({[(2E)-3,7-dimethylocta-2,6-dien-1-yl]amino}methyl)-1λ6-thiolane-1,1-dione
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]benzene-1-sulfonamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(2-{[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
2-[4-(2,3-dihydro-1H-isoindole-2-carbonyl)piperidin-1-yl]acetamide
4-hydroxy-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2-(3-methylphenyl)pyrimidine-5-carboxamide
3-[5-(4-hydroxybutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(4-hydroxypiperidin-1-yl)propan-1-one