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N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-(thiophen-2-yl)acetamide
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4-[(4-methylphenyl)sulfanyl]piperidine
ethyl 4-[(3-fluorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxylate
2-{[6-(propan-2-yl)pyrimidin-4-yl]amino}-1-(thiophen-2-yl)ethan-1-ol
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-3-methylpiperidine-3-carboxamide
(3S,4R)-1-(2-amino-9H-purin-6-yl)-3-benzyl-4-methylpiperidin-4-ol
N-(2,3-dihydro-1H-inden-4-yl)-4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carboxamide
(1s,4s)-4-{4-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
ethyl 1-benzyl-5-[(4-acetamidophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{[4-(2,5-dimethoxybenzoyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
3-{[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}[2-(1H-1,2,4-triazol-1-yl)propyl]amine
2-methyl-7-[4-(1H-pyrazol-4-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[(1-phenylcyclopentyl)methyl]-6-(1,3-thiazol-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-4-(1H-pyrazol-4-yl)quinoline
N-[(3-methoxyphenyl)methyl]-2-methyl-N-(2-methylpropyl)imidazo[1,2-a]pyrimidine-3-carboxamide
1-(2-methylphenyl)-4-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
(2E)-1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-phenylprop-2-en-1-one
N-(oxan-4-yl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
methyl 5-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}furan-2-carboxylate
2-(morpholin-4-ylmethyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)-1,4-oxazepane
N-[(2R,3R)-1'-(2,6-difluorobenzoyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
8-(1-methyl-1H-pyrazole-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 3-[(2-fluoro-5-methoxyphenyl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(3aS,6aS)-2-[5-(1H-1,3-benzodiazol-1-ylmethyl)-1,2-oxazole-3-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-[2-(diethylamino)ethyl]-N-ethyl-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
7-chloro-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}quinoxaline
1-{2-[2-(3-chlorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(propan-2-yl)piperidine-4-carboxamide
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-methoxy-N-methyl-4-oxo-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,4-dihydropyridine-2-carboxamide
N-(2-chloro-3,5-difluorophenyl)-4-cyclopentyl-3-oxopiperazine-1-carboxamide
N-(2-{7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
N-methyl-4-phenyl-N-[1-(2-phenylethyl)piperidin-3-yl]butanamide
2-ethoxy-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-(5-fluoro-2-methylbenzoyl)piperazine-2-carboxylic acid
1-(2-methoxyethyl)-3-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
2-[4-methyl-1-(4-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
6-methyl-2-phenyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-4-amine
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-methyl-4-[2-(methylsulfanyl)ethyl]-5-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}-1,2,3,4-tetrahydropyrimidin-2-one
1-[2-({[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}amino)pyrimidin-4-yl]piperidin-3-ol
1-(4-oxo-4H-chromen-6-yl)-3-[2-(propylsulfanyl)ethyl]urea
N-cyclobutyl-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{4-[(4-fluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol