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N-[2-(furan-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-cyclopropyl-4-methyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-one
1-(3-{[3-(2-oxoimidazolidin-1-yl)phenyl]formamido}propyl)piperidine-3-carboxamide
4-[(2,3-dichloro-6-fluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
1-(3-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-oxopropyl)piperidin-2-one
3-(3-fluorophenoxymethyl)-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidine
2-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-5-phenyl-1,2-oxazole-4-carboxamide
3-(hydroxymethyl)-1-(quinoline-3-carbonyl)piperidin-3-ol
1-(1-aminocyclopropanecarbonyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
N-[(3S,4R)-4-(propan-2-yl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]acetamide
2,4-dimethyl-5-{[2-(3-phenylpyrrolidin-1-yl)ethyl]carbamoyl}-1H-pyrrole-3-carboxylic acid
2-{[4-(2-methoxyphenyl)-5-(3-methyl-1,2-oxazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
9-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-5-methylpyrazine
N-[4-methoxy-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]carbamoyl}amino)phenyl]acetamide
7-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
1-(7-fluoro-4,6-dimethylquinazolin-2-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]piperidin-4-amine
7-[(2-fluorophenyl)methyl]-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-methyl-5-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(4-hydroxyazepan-4-yl)methyl]-2-[4-(hydroxymethyl)phenyl]acetamide
1-[3-(3-chlorophenyl)-3-phenylpropanoyl]-1,4-diazepan-5-one
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-{5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-pyrazol-3-yl}phenol
(1S,5R)-3-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,9aR)-1-{[4-(2-methylpropyl)piperazin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
2-methyl-4-{3-methyl-5-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-1H-1,2,4-triazol-1-yl}pyridine
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-2-(methylamino)pyrimidine-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-(2,3-dimethylphenyl)-N-methylpyridine-3-carboxamide
5-acetyl-N-cyclopropyl-N-(1H-indol-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,9aR)-8-benzoyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-5-phenylpentane-1,5-dione
3-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)-1,3-oxazolidin-2-one
1-[1-(5-cyanopyridin-2-yl)piperidin-3-yl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4,4,4-trifluorobutan-1-one
N-(2-fluorophenyl)-3-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}propanamide
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-(oxolan-3-ylmethyl)piperidine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
2-(2,3-dimethoxyphenyl)-2-[4-(2-methoxyethyl)piperazin-1-yl]acetic acid
4-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperazine-1-sulfonamide
4-(4-chlorophenyl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]butan-1-one
8-methoxy-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
N-[2-(5-chlorothiophen-2-yl)pyridin-3-yl]-2-methylpropanamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
2-(4-methylphenoxy)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione