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1-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
3-cyclopentyl-5-(2,3-dihydro-1,4-benzodioxine-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-{2-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
1-benzyl-N-ethyl-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl[(3-methyl-1H-pyrazol-4-yl)methyl][2-methyl-2-(morpholin-4-yl)propyl]amine
ethyl 1-(oxolane-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-(diethylamino)-3-[4-({[(4-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-(1,3-benzothiazol-2-ylmethyl)-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
methyl 2-[2-(dimethylcarbamoyl)ethyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
6-{1-[(5-chlorofuran-2-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
5-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1H-imidazole-4-carboxylic acid
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)pyridine-2-carboxamide
1-{1-[(4-carbamoylphenyl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-3-carboxamide
N-(2-{2-[4-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)acetamide
(1R,3R,5S)-3-(4-methoxyphenyl)-8-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-8-azabicyclo[3.2.1]octane
N-butyl-3-ethyl-N-(furan-2-ylmethyl)-4-methyl-1H-pyrazole-5-carboxamide
N-[2-(4-fluorophenyl)ethyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
6-chloro-3-(3-hydroxy-2,2-dimethylpropyl)-8-methyl-3,4-dihydroquinazolin-4-one
N-{[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
6-ethoxy-3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-(1H-imidazol-1-yl)acetamide
N-[2-({4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxyphenyl}formamido)ethyl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
4-methoxy-N-{2-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
3-{[2-(2-ethylphenoxy)ethyl](methyl)amino}propane-1,2-diol
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(1H-1,2,4-triazol-1-yl)butanamide
1-(2,6-diaminopyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
9-methyl-3-[4-(trifluoromethyl)pyrimidin-2-yl]-3,9-diazaspiro[5.6]dodecan-10-one
5-{1-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
9-(3-chloro-2-methylbenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carbonyl]piperazin-2-one
5-[(2S)-1-cyclohexanecarbonylpyrrolidin-2-yl]-1-[2-(1H-imidazol-5-yl)ethyl]-3-methyl-1H-1,2,4-triazole
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(1-methyl-1H-imidazol-2-yl)methyl]amine
7-(2,6-dimethoxyphenyl)-9-methoxy-4-(4-methylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[(3-methoxyphenyl)methoxy]-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
(2R)-2-amino-N,4-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pentanamide
N5-cyclooctyl-N3-(furan-2-ylmethyl)-1-(2-methoxyethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
8-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)acetamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[3-(3-fluorophenyl)phenyl]piperidin-4-amine
2-{1-[(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
4-phenyl-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]pyrimidin-2-amine
2-{5-[5-(oxan-2-yl)thiophen-2-yl]-4-phenyl-1H-imidazol-1-yl}ethan-1-ol