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2-(3-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}phenoxy)acetamide
1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-4-(hydroxymethyl)azepan-4-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(4-phenylbutanoyl)piperidine-2-carboxamide
1-(1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}azetidin-3-yl)piperidine
N-{1-[(3-chlorophenyl)methyl]azepan-4-yl}-2-(pyridin-3-yl)acetamide
4-(2-ethylpyridine-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4-chloro-2-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)acetic acid
4-(4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazin-1-yl)-6-methylpyrimidin-2-amine
4-({4-[(3,4-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-3-ethylpiperazin-2-one
methyl 8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
4-(piperidin-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
2-hydroxy-5-{[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]methyl}benzoic acid
N-(2-hydroxyethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-[(4-chlorophenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-[(2R,3R)-2-ethoxy-1'-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-{2-cyclobutanecarbonyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
2-(2,5-dimethylphenoxy)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}propan-1-one
7-fluoro-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
N,N-dimethyl-3-({2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}sulfamoyl)benzamide
3-[(3R,4S)-4-(dimethylamino)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-3-yl]propan-1-ol
N-[4-(2,1,3-benzoxadiazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-(dimethylamino)acetamide
4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-1-(2-methylbutyl)piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1,8-dibenzyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S)-1-(1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)pyrrolidine-2-carboxylate
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-ol
methyl 2-[2-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenoxy]acetate
2-cyclohexyl-5-[1-(6-methoxypyridin-3-yl)-1H-imidazol-2-yl]pyrimidine
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-methoxy-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
N-[4-(3-fluorophenyl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-3-carboxamide
2-{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(2-phenylethyl)piperidin-3-ol
1-methanesulfonyl-N-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-amine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-methoxyphenyl)ethan-1-one
3-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-(propan-2-yl)-5-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
ethyl 3-[(2-fluorophenyl)methyl]-1-[2-(piperidin-1-yl)acetyl]piperidine-3-carboxylate
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(quinoline-3-carbonyl)pyrrolidin-3-yl]urea
(2S)-N-{[1-(dimethylamino)cyclohexyl]methyl}-2-hydroxy-3-phenylpropanamide
N-methyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
N-(2,4-dichloro-3-methylphenyl)-4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-acetamidopropanamide
2-(methoxymethyl)-1-methyl-5-(2-phenylacetamido)-N-[3-(pyridin-3-yloxy)propyl]-1H-1,3-benzodiazole-7-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
7-chloro-2,4-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide