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6-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
N-(1-hydroxy-2-methylpropan-2-yl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl[1-(pyridin-3-yl)ethyl]{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
2-[3-cyclopropyl-5-(2-methanesulfonylethyl)-1H-1,2,4-triazol-1-yl]acetic acid
(1S,5R)-3-benzyl-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
5-(3-fluorophenoxymethyl)-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1H-pyrazole-3-carboxamide
9-(4-fluoro-3-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
(3S,4S)-1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
8-chloro-2-[({[4-(hydroxymethyl)phenyl]methyl}amino)methyl]quinolin-4-ol
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(6-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrrolidine
1-(3-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-one
5-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
3-[(3R,4S)-1-[2-(2,4-dimethoxyphenyl)acetyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
5-[1-(methylsulfanyl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(2S,4S)-N-ethyl-4-[3-(4-methoxyphenyl)propanamido]-1-methylpyrrolidine-2-carboxamide
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
2-[4-(methylsulfanyl)phenyl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-cyclobutanecarbonyl-9-(oxolan-3-ylmethoxy)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)-5-{1-[3-(thiophen-2-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
(3aR,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-methoxypropan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]propan-1-one
1-[1'-(2,4-dimethylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-3-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
1-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxylic acid
2-cyclopentyl-4-[4-(oxolane-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 2-(1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-1H-pyrazol-4-yl}-N-methylformamido)acetate
2-[1-(4-chlorophenyl)piperidin-4-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
3-[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]benzonitrile
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
N-[1-(methoxymethyl)cyclopentyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-cyclopropyl-8-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
3-benzyl-8-{[2-(furan-2-yl)phenyl]methyl}-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(6-methoxypyridin-3-yl)phenyl]butan-1-ol
1-(furan-3-carbonyl)-4-[4-(trifluoromethyl)pyrimidin-2-yl]-1,4-diazepane
2,8-dimethyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)quinoline-4-carboxamide
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[3-(pyridin-3-yl)propyl]acetamide
8-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-2-propyl-N-(1,3-thiazol-2-ylmethyl)-1,3-thiazole-4-carboxamide
6-methyl-2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}pyridine-3-carbonitrile
2-[(5-methylpyrazin-2-yl)methyl]-9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-3-yl)piperazine
3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-ol
ethyl 2-(4-{4-[4-(2,4-dimethylbenzamido)-1H-pyrazol-1-yl]benzoyl}morpholin-3-yl)acetate
N-[(4,6-dimethylpyridin-2-yl)methyl]-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}pyridine-3-carboxylic acid