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1-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)piperidine-4-carboxamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)-1-phenylethyl]amine
1-[4-(dimethylamino)azepan-1-yl]-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
3-[1-(4-methoxypyridine-2-carbonyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
ethyl 4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
methyl[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
8-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-(2-fluorophenyl)-4-[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]piperazine
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-(1H-pyrazol-4-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]prop-2-enamide
3-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-4H-chromen-4-one
4-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
N-(prop-2-en-1-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
methyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(2-hydroxyphenyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]acetamide
6,7-dimethoxy-1-[(4-methylphenyl)methyl]-3-{[(thiophen-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
8-{2-[ethyl(methyl)amino]acetyl}-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3-{4-[2-(1H-imidazol-1-yl)ethyl]piperazine-1-carbonyl}phenyl)-2-methylbutan-2-ol
N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
4-[3-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
[(3S,5R)-1-(2,5-dimethoxybenzoyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-1,3-thiazole-4-carboxamide
1-[4-(aminomethyl)phenyl]-3-[4-(oxolan-2-yl)butyl]urea
1-{[2-({[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
5-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
(3S,4S)-4-(4-fluorophenyl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
1-[4-(4-acetylphenyl)piperazin-1-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propan-1-one
2-ethyl-5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]pyrimidine
N-(1-hydroxypropan-2-yl)-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
N-(2-methyl-1-{7-[2-(phenylsulfanyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)oxolane-3-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(pyrrolidin-1-yl)propyl]-1H-pyrazole-3-carboxamide
2-(methylsulfanyl)-N-[(3R,4S)-4-propyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-(2-hydroxyethyl)-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-(4,4-difluoropiperidin-1-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-[(2,6-difluoro-3-methylphenyl)methyl]-2-(1-methylpiperidin-2-yl)acetamide
(3S,4R)-1-[2-(2-ethylphenoxy)ethyl]-4-methylpiperidine-3,4-diol
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(pyridin-3-yl)acetamide
1-[6-(aminomethyl)-2-methylpyrimidin-4-yl]-4-phenylpiperidine-4-carbonitrile
2-(1H-1,3-benzodiazol-1-yl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
7-(cyclopropylmethyl)-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-[4-(1-benzothiophene-5-carbonyl)piperazin-1-yl]pyrazine
3-methyl-1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazol-5-amine