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1-(2-methylphenyl)-3-(1-{1-[2-(piperidin-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-[(5-chloro-2,4-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)cyclopropanamine
3-(dimethylsulfamoyl)-5-{[(5-ethylfuran-2-yl)methyl]amino}-N-[3-(1H-imidazol-1-yl)propyl]benzamide
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2H-1,2,3-benzotriazol-2-yl)ethan-1-one
2-[(4-chlorophenyl)methyl]-N-[2-(methylamino)ethyl]benzamide
5-methyl-1'-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(3R,5S)-1-benzyl-N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-2-ethyl-6-methyl-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-{5-[1-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]furan-2-yl}benzene-1-sulfonamide
[(1-ethyl-1H-imidazol-2-yl)methyl]({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-cyclopentyl-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)acetamide
(3aR,5S,6S,7aS)-2-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-octahydro-1H-isoindole-5,6-diol
1-(cyclopropylmethyl)-4-[2-(1H-imidazol-2-yl)benzoyl]-2-(propan-2-yl)-1,4-diazepane
[(5-methoxy-1H-indazol-3-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
1-(2-{1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}acetyl)-N,N-diethylpiperidine-3-carboxamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-methylbenzene-1-sulfonamide
4-({1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}methyl)morpholine
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,2-dione
1-(6-ethylpyrimidin-4-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
1-[1-(2-methoxyacetyl)piperidine-4-carbonyl]-4-phenylpiperidine-4-carbonitrile
(1S,5R)-3-benzoyl-6-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-[3-(propan-2-yloxy)phenyl]pyridine-3-carbonitrile
1-[2-(4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}phenoxy)ethyl]-1H-imidazole
N-[4-(furan-2-yl)butan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N,N-dimethyl-3-({[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]carbamoyl}amino)benzamide
3-[(dimethylamino)methyl]-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-3-ol
(2S,4R)-4-amino-1-(2-ethoxybenzoyl)-N-methylpyrrolidine-2-carboxamide
1-[2-methoxy-5-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
N-(2,3-dihydro-1H-inden-1-yl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-(3-hydroxyphenyl)-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
4-phenyl-N-(1,3,4-thiadiazol-2-yl)azepane-1-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)acetamide
4-{[(3-fluoro-2,4-dimethylphenyl)methyl](methyl)amino}-2-methylbutan-2-ol
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3,4-difluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 4-({7-oxo-4-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-1,4-diazepan-1-yl}methyl)benzoate
methyl 3-acetamido-1-(3-methylbutyl)-5-({[4-(methylsulfanyl)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl (2S,4R)-1-{4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanoyl}-4-hydroxypyrrolidine-2-carboxylate
9-[2-hydroxy-4-(methylsulfanyl)butanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
3-phenoxy-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(5-methoxyfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(6-chloropyridin-3-yl)-4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
6-chloro-N,2-dimethyl-N-[1-(pyridin-2-yl)propyl]imidazo[1,2-a]pyridine-3-carboxamide
2-(oxolane-2-carbonyl)-8-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
7-chloro-N-ethyl-N-[(2-fluorophenyl)methyl]-1-methyl-1H-indole-2-carboxamide
(4aR,7aS)-1-ethyl-4-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione