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8-({[2-(4-fluorophenyl)ethyl]carbamoyl}methyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[2-(1H-imidazol-1-yl)ethyl]-N,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
1-[(2-chloro-4-fluorophenyl)methyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
(4aR,8aS)-1-cyclopropanecarbonyl-6-(2-methylpropyl)-decahydro-1,6-naphthyridine
(5-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}furan-2-yl)methanol
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2,2-diethylcyclopropanecarbonyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[3-(5-methyl-1H-pyrazol-1-yl)propyl]-3-phenylpiperidine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-5-methoxy-3-methyl-1H-indole-2-carboxamide
1-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
{[4-(6-cyclopropylpyrimidin-4-yl)phenyl]methyl}dimethylamine
5-(5-aminopyridin-3-yl)-6-methyl-1,3-benzothiazol-2-amine
1-[2-(2-methoxyethoxy)phenyl]-3-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]urea
1-(2-{[2-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)piperidin-2-one
1-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethoxy)piperidine
(1S)-2-(1H-imidazol-4-yl)-1-{1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethan-1-amine
2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)phenoxy]ethan-1-ol
methyl 5-({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}amino)-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(2-methoxyphenyl)ethyl]propanamide
2-{[6-(quinolin-6-yl)pyrazin-2-yl]sulfanyl}acetic acid
5-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3,5-dimethyl-4,5-dihydro-1,2-oxazole
N-[(2S)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
4-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
N-[(5-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}bis(1,3-oxazol-4-ylmethyl)amine
1-(2-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
4-{[({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]methyl}hepta-1,6-dien-4-ol
(1S,5R)-6-[(5-chlorothiophen-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}pyridine
methyl 1-[5-methanesulfonamido-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-4-carboxylate
1-[1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(4-methylphenyl)methyl]piperidin-3-yl]propanoate
3-cyclohexyl-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
5-propyl-N-[2-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
ethyl 2-({2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]phenyl}amino)acetate
2-ethoxy-5-(2-{[1-(1H-imidazol-2-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
4-(2,3-dimethoxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-4-phenylbutane-1,2-dione
4-ethyl-3-{[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(naphthalen-2-yloxy)propanamide
methyl 5-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)furan-2-carboxylate
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}propanamide
1-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
4-(1H-indole-6-carbonyl)-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-{4-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]quinazolin-2-yl}ethan-1-amine
4-(4-{[ethyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]propan-1-one
methyl 2-{8-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-methyl-2-(morpholin-4-yl)propyl]benzamide