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3-(dimethylamino)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
3-(3-fluorophenyl)-4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
ethyl 2-({3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}amino)acetate
1-[(2,6-difluoro-4-methoxyphenyl)methyl]-3-methoxypyrrolidine
5-(2-methoxypyridin-3-yl)pyridin-2-amine
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N,N-diethyl-1-[(1s,4s)-4-(2-phenoxyacetamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)carbamoyl}amino)phenyl]acetamide
2-tert-butyl-4-hydroxy-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}methyl)piperidin-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}acetamide
methyl 3-(furan-2-amido)-1-methyl-5-{[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-ethyl-4-(pyrrolidin-1-ylmethyl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]furan-2-carboxamide
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-2-ol
1-[(2-fluorophenyl)methyl]-N-methyl-N-(2-phenoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-methylazepan-4-ol
1-{3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
N-[(1-benzylpyrrolidin-3-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(4-methylphenyl)-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
6-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-2,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
7-(3-propyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(5-ethylthiophene-3-carbonyl)piperidine
1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
3-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(2,4-difluorophenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
[(3-chloro-4-methoxyphenyl)methyl](1,4-dioxan-2-ylmethyl)methylamine
ethyl 1-(cyclopropylmethyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
5-chloro-1,3-dimethyl-4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
2-(1H-pyrazol-1-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-ol
N,N-dimethyl-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzamide
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[4-(oxolan-2-yl)butyl]acetamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-(methylsulfanyl)benzamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
methyl 2-{3-oxo-1-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperazin-2-yl}acetate
1-(6-cyanopyridin-3-yl)-3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-methylurea
2-({[1-(methoxymethyl)cyclobutyl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2,2-diphenyl-1-[4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
(3R,5S)-N-[2-(dimethylamino)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1-(2-phenylethyl)piperidine-3-carboxamide
1-methyl-4-(4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)-1,4-diazepane
3-(6-hydroxy-1,4-oxazepane-4-carbonyl)-1-methyl-1,2-dihydroquinoxalin-2-one
2-{[(3,4,5-trimethoxyphenyl)methyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one