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4-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(2-methylphenyl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
N-(2H-1,3-benzodioxol-5-yl)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
1-(2-methoxyethyl)-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazine
N-[(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]-1H-indole-2-carboxamide
2-amino-6-(1-ethyl-1H-indol-3-yl)-4-(pyridin-4-yl)pyridine-3-carbonitrile
(2-methoxyethyl)[(6-methoxypyridin-3-yl)methyl][(4-methylphenyl)methyl]amine
5-cyclopropyl-N-[2-(5-methylfuran-2-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[5-(2-hydroxy-3-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-7-methyl-1-benzofuran-2-carboxamide
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
4-{5-methyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}-1,4-diazepane-1-carbaldehyde
14-(pyrimidin-5-yl)-2,17-diazatetracyclo[9.8.0.03,8.013,18]nonadeca-1(19),3(8),4,6,11,13(18)-hexaen-16-one
2-(3,4-dimethoxyphenyl)-1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
(4aR,7aS)-1-(2-methoxyacetyl)-4-(1,2,4-oxadiazol-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-1,3-benzothiazole
6-(3,4,5-trimethoxyphenyl)-3H-imidazo[4,5-b]pyridine
(2R,6R)-10-methoxy-4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-phenoxy-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
(2S,4R)-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-({4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
4-{[3-(1-phenoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
3-[5-(5-methoxypentyl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
1-(5-methanesulfonyl-2-methylphenyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
(4aS,7aR)-1-cycloheptanecarbonyl-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-methyl-5-(methylcarbamoyl)phenyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-(2-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)-1,3-thiazole
N-{[6-(2-chloro-4-fluorophenyl)pyridin-3-yl]methyl}acetamide
2-[(2-amino-6-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrimidin-4-yl)amino]ethan-1-ol
N-[4-(propan-2-yl)phenyl]-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-amine
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-methoxypiperidine
2-[3,5-dimethyl-4-(2-methylphenyl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-indazol-3-yl)acetamide
3-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1-[(5-methyl-1H-pyrazol-3-yl)methyl]urea
2-(dimethylamino)-7-[(2R)-pyrrolidine-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{4-[(2-chlorophenyl)methyl]-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[4-(2,6-dimethoxypyridine-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
6-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
4-(2-phenylquinazolin-4-yl)-1,4-oxazepan-6-ol
2-(1H-imidazol-4-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
2-(3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenoxymethyl)pyridine
(3R,4R)-3-cyclopropyl-1-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}-4-methylpyrrolidin-3-ol
3-[4-(3-methyl-3-phenylpiperidin-1-yl)piperidine-1-carbonyl]pyridine
2-(4-{[methyl({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl})amino]methyl}piperidin-1-yl)ethan-1-ol
7-(3-chlorophenyl)-4-(4-methylpyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
4-[(3-phenoxyphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,5R)-5-(cyclopropylcarbamoyl)-1-(2,2-diphenylethyl)piperidine-3-carboxylic acid
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-methoxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}propanamide