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N-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
1-[1-(pyrazin-2-yl)piperidin-3-yl]-3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]urea
3-(2,5-dimethoxyphenyl)-N-(1,2,3-thiadiazol-5-yl)pyrrolidine-1-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-4-acetamido-2-methylbenzamide
2-(azepan-1-yl)-N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)acetamide
4-methyl-2-oxo-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-7-thia-2,5-diazatricyclo[6.4.0.02,6]dodeca-1(12),5,8,10-tetraen-11-amine
9-benzoyl-4-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane
(3R)-3,4,4-trimethyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-[(3S,4R)-1-[(5-chlorothiophen-2-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-[(3,4-dimethoxyphenyl)methyl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]-6-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
2-[3-(2-phenylethyl)-5-{[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazol-1-yl]pyridine
N-[1-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
2-[2,4-dioxo-1-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
1-{3-methyl-5-[4-(methylsulfanyl)phenyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-cyclopropyl-1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-butanamido-N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]benzamide
methyl 5-{[(4-ethylphenyl)methyl]amino}-1-(2-methylpropyl)-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,4S)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-propylpyrrolidine-3-carboxylic acid
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methoxyphenyl)methyl]acetamide
3-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
5-fluoro-6-methyl-2-(4-{[methyl(2-phenylethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-(1-{4-[6-(2-methyl-1H-imidazol-1-yl)pyridazin-3-yl]phenyl}ethyl)morpholine
1-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperidine-4-carbonitrile
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-3-methoxybenzamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
3-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carboxamide
N-{[4-(morpholin-4-yl)phenyl]methyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
3-{[1-(4-fluorophenyl)-2-hydroxyethyl]sulfamoyl}-N-propylbenzamide
N-[(2-chloropyridin-3-yl)methyl]-N,6-dimethyl-2-(pyridin-3-yl)pyrimidin-4-amine
5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}acetamide
5-ethyl-N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1,2-oxazole-3-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
1-(4-chloro-3-fluorophenyl)-3-[2-(1-hydroxycyclopentyl)ethyl]-3-methylurea
3-[2-oxo-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethyl]-1,3-oxazolidin-2-one
1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
[2-({4-[(5-chlorofuran-2-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-methyl-5-phenyl-N-(pyrimidin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-[(3-hydroxyphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[1'-(2-ethylpyrimidine-5-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
2-{2-[(4-hydroxypiperidin-1-yl)methyl]phenyl}-6-propyl-3,4-dihydropyrimidin-4-one
N-(1H-1,3-benzodiazol-2-yl)-2-({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)acetamide
methyl (2S)-2-[(benzylsulfamoyl)amino]-4-methylpentanoate
methyl 8-(furan-2-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate