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1-[3-(azepan-1-yl)propyl]-3-(1H-1,3-benzodiazol-5-yl)-1-methylurea
2-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-6-methoxyphenol
2-[3-({5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)piperidin-1-yl]ethan-1-ol
3-(5-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}thiophen-2-yl)prop-2-yn-1-ol
1-{2-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
{2-fluoro-5-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]phenyl}methanol
3-methyl-6-{5-[(propylsulfanyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-(1-benzylpiperidin-4-yl)-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[2-(hydroxymethyl)phenyl]-2-(1,2-oxazol-5-yl)phenol
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2-methoxyphenyl)ethan-1-one
4-{5-[2-(2-oxopyrrolidin-1-yl)ethyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-3-yl}benzamide
5-methyl-1'-(2-propyl-1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl][(1-ethyl-1H-indol-4-yl)methyl]methylamine
{5-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]furan-2-yl}methanol
1-cyclohexyl-N3-[(3,5-dimethoxyphenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
{[4-(6-methoxypyrimidin-4-yl)-1,4-oxazepan-6-yl]methyl}dimethylamine
4-[(2-fluoro-5-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-methoxy-N,3-dimethyl-1H-indole-2-carboxamide
3,5-dimethyl-N-{3-methyl-1-[7-(thiophene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
1-(1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3-[4-(trifluoromethyl)benzoyl]piperidine
8-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(pyridin-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
2,6-dimethyl-5-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-1-phenylcyclopropane-1-carboxamide
{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(3R,4R)-1-(4-amino-6,7-dimethoxyquinazolin-2-yl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
3-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
4-methoxy-N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
(5S)-5-({[(3-methyl-1,2-oxazol-5-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
8-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1-methyl-1H-pyrazole-5-carboxamide
2-amino-6-(1H-indol-3-yl)-4-(1-methylpiperidin-4-yl)pyridine-3-carbonitrile
N-(1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl)methanesulfonamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
N-cyclohexyl-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-benzyl-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-{2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(5-methylthiophen-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-5-carboxamide
1-cyclopentyl-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
2-[N-(3-methylphenyl)methanesulfonamido]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)methanesulfonamide
(3aS,7aR)-5-methyl-2-[3-(thiophen-3-yl)propanoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[(4-chlorophenyl)methyl]-N-methyl-N-(quinolin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl](oxolan-2-ylmethyl)amine
ethyl 4-[(2-chlorophenyl)methyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidine-4-carboxylate