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2-methyl-1-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]propan-1-one
8-[(4-{2-[3-(morpholin-4-ylmethyl)phenoxy]ethyl}piperazin-1-yl)sulfonyl]quinoline
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N,4-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1,2,3-thiadiazole-5-carboxamide
(1S,5R)-3-(2-methyl-1H-pyrrole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-3-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-fluoro-4-methoxybenzoyl)-1-[4-(propan-2-yloxy)benzoyl]piperidine
methyl (2S,4R)-1-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-(dimethylamino)pyrrolidine-2-carboxylate
N-[(2S)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
N-({7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
N,N-diethyl-1-({1-[2-(2-methylphenyl)acetyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
2-(3-fluoro-5-methylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
N-(piperidin-4-ylmethyl)-2-(4-propanoylphenoxy)acetamide
2-{[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(cyclopropylmethyl)sulfanyl]-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(3-hydroxypropyl)-9-[2-(phenylsulfanyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6,7-dimethoxy-3-(thiophen-3-ylmethyl)-3,4-dihydroquinazolin-4-one
6-methyl-3-{[methyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
N-methyl-N-(oxan-2-ylmethyl)-3-sulfamoylbenzamide
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
4-[2-(piperidine-1-carbonyl)phenoxy]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine
2-[1-({1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[3-(trifluoromethyl)phenyl]urea
N-[(3S,4R)-1-(7-methoxy-4-methylquinolin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-{[(4-methylphenyl)methyl]amino}benzamide
1-[5-methoxy-2-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-{3-[2-(8-fluoroquinolin-2-yl)-1H-imidazol-1-yl]piperidin-1-yl}-2-methylpropan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-(5-chloropyridine-3-carbonyl)-4-cyclohexyl-1,4-diazepane
1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
1-{2-[1-(cyclohexylmethyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
(3R,5S)-N-[3-(dimethylamino)propyl]-5-[(4-methylpiperazin-1-yl)methyl]-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
N-[(1-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-3-yl)methyl]acetamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-5-(methoxymethyl)thiophene-2-carboxamide
2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-N-[(2-methoxyphenyl)methyl]acetamide
3-({1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
1-[5-(propan-2-yl)thiophene-3-carbonyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
1-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazole
2-methyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}quinoline-4-carboxylic acid
3-(4-cyano-4-phenylpiperidine-1-carbonyl)-N,N-dimethylpiperidine-1-carboxamide
N-butyl-N-[(3-chlorophenyl)methyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(1-cyclopentanecarbonylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]-4-methoxybenzamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[(methylsulfanyl)methyl]-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyridine
(2R,3R)-3-amino-1'-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{[(5-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol