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2-[3-(5-methylfuran-2-yl)-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
(2S,4R)-4-amino-N-methyl-1-{[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]sulfonyl}pyrrolidine-2-carboxamide
2,4,5-trimethyl-6-(2,3,4-trimethoxyphenyl)pyrimidine
4-[(5-ethylpyridin-2-yl)methyl]-3-(4-fluorophenyl)piperazin-2-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-hydroxybutanamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
4-(1H-imidazol-2-yl)-1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine
(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
(2R)-1-({4-[(2H-1,3-benzodioxol-5-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide
2-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-dihydroisoquinolin-1-one
methyl 6-benzoyl-2-[(3-fluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(1-ethyl-1H-imidazol-2-yl)-1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidine
3-[(3R,4S)-1-(8-chloroquinolin-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
7-(2-methoxyacetamido)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
3-(3-{1-[2-(piperidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine
1-[2-(1H-imidazol-4-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
5-[2-(methylsulfanyl)phenoxymethyl]-3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,2-oxazole
8-chloro-2-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
1-{4-[(cyclopropylcarbamoyl)methyl]phenyl}-5-oxopyrrolidine-3-carboxylic acid
(3S,5S)-1-cyclobutanecarbonyl-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(6-methylpyridazin-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-chloro-N-(2-methoxyethyl)-4-({1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}oxy)benzamide
N-[1-(2-methoxyphenoxy)propan-2-yl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2S)-2-amino-N-[1-(4-methoxyphenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]butanamide
N-[2-(7-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
2-amino-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)pyridine-4-carboxamide
1-[3-(4-methylpiperazin-1-yl)propyl]-3-(6-phenoxypyridin-3-yl)urea
(2S,4R)-4-amino-1-(4-chloro-2-hydroxybenzoyl)-N-ethylpyrrolidine-2-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
3-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
2,4-dimethyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(pyridin-4-ylsulfanyl)acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-methylthian-4-amine
N-butyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methylpiperidine-3-carboxamide
2-[3-({[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenoxy]ethan-1-ol
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}acetamide
1-{4-[4-(5-ethyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]phenyl}ethan-1-one
7-cyclohexyl-2-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2-chloro-6-fluorophenyl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-cyclohexanecarbonyl-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
N-(2-ethylphenyl)-3-({5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)propanamide
2-(pyridin-3-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
methyl (2S,4R)-4-(3-chlorobenzamido)-1-[(2-ethoxyphenyl)methyl]pyrrolidine-2-carboxylate
2-[4-(benzyloxy)piperidin-1-yl]-1,3-thiazole-4-carboxamide
7-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-2-oxa-7-azaspiro[4.5]decan-8-one
1-({5-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
N-[(3S,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-7,8-dimethyl-3,4-dihydroquinazolin-4-one
methyl 2-methoxy-4-[(thiomorpholine-4-carbonyl)amino]benzoate
(2E)-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(4-methoxyphenyl)prop-2-enamide