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6-{4-[1-(morpholin-4-yl)ethyl]phenyl}-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidin-4-amine
2-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-7-ethyl-2,7-diazaspiro[4.4]nonane
2-[1-(2,2-dimethylpropyl)-4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
(2S,4R)-4-amino-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-methyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-3-[(pyridin-2-ylmethyl)amino]benzamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
(3S,4S)-4-cyclopropyl-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]pyrrolidine-3-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(propan-2-yl)benzenesulfonamido]acetic acid
4-(2,4-dimethoxyphenyl)-3-methylpyridine
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[2-(1-propylpiperidin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
ethyl 4-{6-methyl-3-[({spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}amino)methyl]quinolin-2-yl}piperazine-1-carboxylate
1-(2H-1,3-benzodioxol-5-yl)-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazole
4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-N,N-dimethylpiperazine-1-sulfonamide
3-(1H-1,3-benzodiazol-1-yl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
1-[2-(dimethylamino)ethyl]-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(3aS,6aR)-5-(1,3-benzothiazol-2-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-{5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}morpholine
4-[4-(2,2-dimethylpropyl)piperazin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-(pyridin-3-yl)ethan-1-one
N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(pyrimidin-4-yl)piperidine-1-carboxamide
2-methoxy-5-({4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)pyridine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]cyclohexanecarboxamide
(3S,4S)-1-(3-methylpyridine-2-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
ethyl 4-({4-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-[(2-methoxyethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
methyl 2-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
methyl 3-[(2-carbamoylmorpholine-4-carbonyl)amino]-4-methylbenzoate
5-(oxolan-2-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}thiophene-2-carboxamide
3-(2-chlorophenyl)-3-phenyl-1-(pyrrolidin-1-yl)propan-1-one
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-3-fluorobenzamide
1-[2-(4-hydroxyphenyl)ethyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
3-methyl-7-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethyl-2,6-dimethylpyrimidin-4-amine
1-({4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}methyl)pyrrolidine
3-({4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}methyl)piperidin-3-ol
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-methyl-3-(morpholine-4-carbonyl)-N-(2-phenylethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(2-methoxyphenyl)-N-(2-methyl-2H-1,2,3-benzotriazol-4-yl)piperidine-1-carboxamide
3-(4-methylpiperidine-1-carbonyl)-5-(4-phenylazepane-1-carbonyl)-1-(propan-2-yl)-1,4-dihydropyridin-4-one
1-(4-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(5S,9aS,9bS)-2-(1-methylpiperidin-4-yl)-5-(naphthalen-1-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1R,2S)-N1-(prop-2-en-1-yl)-N2-[2-(1-propylpiperidin-4-yl)ethyl]cyclohexane-1,2-dicarboxamide
7-[(3-methylphenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
6-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2,3-dimethylquinoxaline
5-{[(2,6-difluoro-3-methylphenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[(6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-3-yl)methyl]morpholine
2-(2,3-dihydro-1H-inden-1-yl)-N-(1,2-oxazol-3-ylmethyl)acetamide