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N-ethyl-N,3,6-trimethyl-2-[2-(pyridin-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-6-cyclopropylpyrimidin-4-amine
3-(2-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,3-diazinane-2,4-dione
N-[1-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-3-yl]-N-ethylacetamide
(3S,4R)-4-methyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine-3,4-diol
ethyl 1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-5-(2,6-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
7-[(3,4-difluorophenyl)methyl]-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-hydroxy-N-methyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
4-{1-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]piperidin-3-yl}benzoic acid
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]pyridine-4-carbonitrile
(4aS,7aR)-1-(furan-3-ylmethyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-cyclohexyl-5-(4-oxo-4-phenylbutyl)-1H-1,2,4-triazol-3-yl]acetamide
4-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 6-benzoyl-2-(benzylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)methyl]acetamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-(pyridin-2-ylmethyl)-5-(pyrrolidine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{4-[2-(cyclopropylcarbamoyl)ethyl]phenyl}-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
1-methyl-N-[3-methyl-2-(pyrrolidin-1-yl)butyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)pyrazine-2-carboxamide
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(dimethylamino)ethyl]-2-methoxy-N-[(2-methylphenyl)methyl]acetamide
8-cyclopropanecarbonyl-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]-6-methylpyridine-3-carbonitrile
2-tert-butyl-4-hydroxy-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrimidine-5-carboxamide
(2R,6R)-4-cyclopentanecarbonyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-(2-methoxyphenyl)-2-methyl-1-(pyridin-4-yl)piperazine
N-ethyl-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]pyrrolidine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperazine
N-ethyl-2-{4-[(5-propylfuran-2-yl)methyl]piperazin-1-yl}acetamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[(4aR,8aS)-6-(4-phenylbutanoyl)-decahydro-1,6-naphthyridine-1-carbonyl]-1,2-dihydrophthalazin-1-one
1-(2-methylpropyl)-4-[1-(piperidine-1-sulfonyl)pyrrolidin-3-yl]piperidine
2-methyl-6-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
N-{1-[(3,4-dimethoxyphenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
2-(1-butyl-1H-pyrazol-4-yl)-N-ethyl-N,3,6-trimethylquinoline-4-carboxamide
N-[(4-ethylphenyl)methyl]-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
3-(3-methylbut-2-en-1-yl)-1-{[4-(methylcarbamoyl)phenyl]methyl}piperidine-3-carboxylic acid
3-(2,5-dimethylphenyl)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]urea
1-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-3-propylurea
(1R,3S)-7-(6-aminopyridine-3-carbonyl)-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
5-(2-methylphenyl)-2-(pyridin-4-yl)-4-[1-(thiophen-2-ylmethyl)piperidin-3-yl]pyrimidine
1-methyl-4-[1-(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)ethyl]piperazine