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[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methanol
2-[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]-N-[1-(4-methylphenyl)ethyl]acetamide
1-(2-ethoxyethyl)-4-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperazine
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}amine
(2S,4R)-4-amino-1-[3-(2-methoxyphenoxy)propyl]-N-methylpyrrolidine-2-carboxamide
6-({2-cyclobutyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-[(4-chlorophenyl)methyl]-3-oxo-N-phenyl-2,8-diazaspiro[4.5]decane-8-carboxamide
3-[6-(dimethylamino)pyrazin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-(1-propylpiperidin-4-yl)imidazolidine-2,4-dione
methyl (2S,4R)-1-benzyl-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
1-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)propan-1-ol
N-(3-chloro-4-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}phenyl)acetamide
(4aS,8aR)-6-[5-(ethylsulfanyl)thiophene-2-carbonyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
6-(adamantane-1-carbonyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
(2R,6S)-1-{imidazo[1,2-a]pyrimidin-6-ylmethyl}-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
6-fluoro-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
5-(2-fluorophenoxymethyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
1-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
7-chloro-4-[4-(3-methoxypropyl)piperazine-1-carbonyl]-2-methylquinoline
N-(3-hydroxypropyl)-4-(5-methylfuran-2-yl)-N-(pyridin-4-ylmethyl)benzamide
[5-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)-2-ethoxyphenyl]methanol
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-(oxan-4-yl)butanamide
2-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
N-[1-(methoxymethyl)cyclopentyl]-N'-(4-methylphenyl)ethanediamide
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
1-methyl-4-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepane
6-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]-7-methyl-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
1-[(3S)-3-aminopiperidin-1-yl]-4-(4-chlorophenyl)butan-1-one
4-{5-[2-(cyclohex-1-en-1-yl)acetyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
[(4-methoxy-2,5-dimethylphenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
1-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(2-methoxyethyl)piperazine
2-methoxy-N-({5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-[1-(1-ethylpiperidin-3-yl)pyrrolidin-3-yl]-N-methylacetamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-{2-[1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
3-{1-butyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
(3S)-1-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-N,N-dimethylazepan-3-amine
4-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-3-yl)pyrimidine
3-ethoxy-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N,5-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{1-[(1-benzyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}pyridine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-propylpyrrolidin-3-yl]-2-hydroxyacetamide
{4-[(2-chlorophenyl)methyl]-1-(1-phenylpiperidin-4-yl)piperidin-4-yl}methanol
1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-[2-(2-fluorophenyl)ethyl]-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
2-cyclopentyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide