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2-{2-[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]ethyl}-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
2-{4-[2-(dimethylamino)-2-(2-methylphenyl)acetamido]piperidin-1-yl}acetic acid
ethyl 1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
4-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)-1,4-oxazepane
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
9-[3-(pyridin-3-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)azepan-2-one
2-(2-fluorophenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(1H-pyrrole-2-carbonyl)piperidin-4-ol
ethyl 4-(7-chloro-3-{[N-cyclopropyl-1-(5-methylthiophen-2-yl)formamido]methyl}quinolin-2-yl)piperazine-1-carboxylate
1-methyl-2-(1-methyl-1H-imidazol-2-yl)-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propanamidobenzamide
5-(2-chloro-4-fluorophenoxymethyl)-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-(furan-2-yl)-1-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-phenylpropan-1-one
2-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2S)-1-(5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-chloro-3-(1H-imidazol-2-yl)-1-methyl-1H-indazole
1-(cyclohex-1-ene-1-carbonyl)-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyridin-3-yl)ethan-1-one
3-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[1-(4-methylpyridin-2-yl)propyl]-2-(4-propanoylphenoxy)acetamide
5-acetyl-2,4-dimethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-pyrrole-3-carboxamide
1-{4-[(3,5-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
4-(2-methoxyethyl)-11-({[4-(trifluoromethoxy)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-methyl-7-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(4-{imidazo[1,2-b]pyridazine-3-carbonyl}morpholin-3-yl)acetic acid
methyl 6-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(3,3-dimethylbutyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
(4aS,8aR)-1-(3-methylbutyl)-6-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-decahydro-1,6-naphthyridin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-methoxybenzamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2S)-2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxypropanamide
ethyl 1-(cyclopropylmethyl)-5-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(3R,4R)-1-[(3-chloro-4-methoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
1-methyl-4-{[methyl({[1-(piperidin-1-yl)cyclohexyl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile
1-[7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]piperidine-3-carbonitrile
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{[4-(propan-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-formyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
1-[(3,4-dimethylphenyl)methyl]-4-[2-(thiophen-3-yl)acetyl]piperazin-2-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine-3-carboxylate
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-2-carboxamide
1-[4-(cyclopropylmethyl)piperazin-1-yl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-(2-methylpropyl)-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one