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(3S,4S)-1-{[2-(benzyloxy)phenyl]methyl}-4-(dimethylamino)pyrrolidin-3-ol
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
3-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propanamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
3-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(2,2-dimethylpropyl)piperazin-2-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
4-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1,2,3-thiadiazole-5-carboxamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
3-{[1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazol-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-{[4-(methylsulfanyl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-cyclopentyl-4-(2,3-dihydro-1H-isoindole-2-carbonyl)pyrrolidin-2-one
N-[(1S,2R)-2-aminocyclobutyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(1-ethyl-5-oxopyrrolidin-3-yl)-3-[(2-hydroxyethyl)(methyl)sulfamoyl]benzamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
8-methoxy-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]quinoline
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-{[1-(morpholin-4-yl)cycloheptyl]methyl}pyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-yl)-3-(2-methoxyethyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
3-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
2-benzyl-N-[3-(pyridin-3-yloxy)propyl]-1,3-benzoxazole-5-carboxamide
N-cyclopropyl-1-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3-{[3-(pyridin-3-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
2-[1-(furan-2-ylmethyl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-yl]ethan-1-ol
2-[2-(4-fluorophenoxy)ethyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 6-[4-(4-chlorophenoxy)piperidin-1-yl]pyrimidine-4-carboxylate
(3R,4S)-4-(3-methoxyphenyl)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-amine
3-{5-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-{2-[4-(dimethylamino)phenyl]ethyl}-2-[methyl(piperidin-4-yl)amino]acetamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]piperidine-3-carboxamide
(2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
1-[(2-chlorophenyl)methyl]-N-[2-(1H-indol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[(3S,5R)-5-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidine-3-carbonyl]morpholine
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
ethyl 4-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylate
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-[(3-fluorophenyl)methyl]morpholine
4-(4-methyl-1H-pyrazol-1-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine-4-carboxylic acid
2-(4-methylpiperidin-1-yl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-2-one
2-(4-chlorophenyl)-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]acetamide
2-[(3,5-difluorophenyl)methyl]-8-methyl-2,8-diazaspiro[4.5]decan-3-one
N-[(2-chloropyridin-3-yl)methyl]-N,8-dimethyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(propane-2-sulfonyl)piperidine
2-amino-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
3-[2-(furan-2-yl)-1H-imidazol-1-yl]-4-hydroxybenzonitrile
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)propanamide
2-[(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)formamido]-N-(propan-2-yl)acetamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(2,5-dimethoxyphenyl)propanamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide