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methyl (2S)-2-{1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-N-methylformamido}propanoate
2-ethyl-N,4-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,3-oxazole-5-carboxamide
1-{5-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-6-methylpyridine-2-carboxamide
N-methyl-N-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)methanesulfonamide
methyl 5-{[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-phenylpiperidine
methyl 3-[2-(2-fluorophenyl)acetyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2,6-dimethyl-8-(4-{4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)octan-2-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-3-carboxamide
2-[3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-6-methyl-3,4-dihydropyrimidin-4-one
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-[(4-methylphenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
1-methyl-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-pyrazole
N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-[1-({3-[1-(dimethylamino)ethyl]phenyl}methyl)piperidin-4-yl]piperidin-4-ol
N-[2-(1H-imidazol-4-yl)ethyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(3-methylphenoxy)-1-(thiophen-2-ylmethyl)azetidine
2-(2-methoxyethyl)-6-[4-(2-phenylethyl)piperidine-1-carbonyl]-1,3-benzoxazole
1-(2-{[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl](methyl)amino}ethyl)piperidin-2-one
3-(3-fluorophenyl)-4-{5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazin-2-one
(1S,5R)-6-[(5-methylfuran-2-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2-chloro-6-methylphenoxy)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]propan-1-one
2-[N-(3-methylphenyl)methanesulfonamido]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]acetamide
2-[4-(2,6-dimethylpyridin-4-yl)phenyl]-2-methylpropanenitrile
N-[(7-{2-[4-(methylsulfanyl)phenyl]acetyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(methylamino)-1,3-thiazole-4-carboxamide
3-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methyl-N-(oxan-4-yl)acetamide
N-[(2-methoxyphenyl)methyl]-2-oxo-N-(prop-2-en-1-yl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
ethyl 2-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}acetate
1-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-(1H-indazol-5-yl)urea
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-(4-fluorophenyl)-1,4-diazepane
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
4-methyl-2-(4-methylpiperazin-1-yl)-N-[(2S)-oxolan-2-ylmethyl]pyrimidine-5-carboxamide
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-propylpiperidin-4-yl]acetate
(1S,5R)-3-(3-cyclopentylpropanoyl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-methoxy-2-methylpropanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
1-({4-methyl-5-[1-(pyridazin-3-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-(2-chloro-4-fluorophenyl)-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-4-(pyridin-2-yl)pyrimidin-2-amine
N-(1,3-dihydroxypropan-2-yl)-2-(phenylamino)pyrimidine-5-carboxamide
3-{[4-(1H-imidazol-1-yl)phenyl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
dimethyl[1-(pyridin-2-yl)-2-(4H-1,2,4-triazol-4-yl)ethyl]amine