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N-butyl-1-(furan-2-ylmethyl)-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
(2S,4S)-4-amino-N-methyl-1-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]pyrrolidine-2-carboxamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1,3-oxazole-4-carboxamide
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
2,6-dimethyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,4-dihydropyridin-4-one
3-(3-{[ethyl(4-hydroxybutyl)amino]methyl}-1H-indol-1-yl)propanamide
4-(5-fluoro-2-methoxybenzoyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-N,N-dimethylpiperazine-1-carboxamide
N-methyl-3-(1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)ethyl]benzamide
4-{1-[1-(propane-1-sulfonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(thiophen-3-ylmethyl)amine
4-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(3-methylphenyl)phenyl]piperidine-1-carboxamide
1-(3,5-dimethyl-1H-indole-2-carbonyl)-4-[(dimethylamino)methyl]azepan-4-ol
4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-2-(thiophen-2-yl)-1,3-thiazole
2-(4-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-3H,4H,5H,7H-thieno[3,4-d]pyrimidin-4-one
ethyl 3-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]carbamoyl}amino)propanoate
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methoxybenzamide
N-[(3R,4S)-4-cyclopropyl-1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]-3-hydroxypropanamide
3-methanesulfonamido-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]propanamide
2-({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
3-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
4-{1-[3-(methylsulfanyl)propanoyl]piperidin-3-yl}benzoic acid
ethyl 1-[2-(1H-1,3-benzodiazol-1-ylmethyl)-1,3-oxazole-4-carbonyl]piperidine-4-carboxylate
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-(2-methylphenyl)-3-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)formamido]propanamide
N-ethyl-N-(pyridin-4-ylmethyl)-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-amine
1-{4-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-oxobutyl}piperidin-2-one
N-(oxan-2-ylmethyl)-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
methyl 5-[(1-benzofuran-2-ylmethyl)amino]-1-benzyl-3-cyclopropaneamido-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,3R)-3-hydroxy-2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}butanamide
5-(morpholin-4-yl)-2-(2-oxo-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethyl)-2,3-dihydropyridazin-3-one
1-[2-(2-hydroxyethyl)piperidin-1-yl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-(1-benzyl-4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
(4aS,7aR)-1-(2-fluorobenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
5-ethyl-4-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]pyrimidin-2-amine
methyl[(3-methylpyridin-4-yl)methyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
1-[3-(morpholin-4-yl)propyl]-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)piperidin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)acetamide
2-(pyridin-3-yl)-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-5,6,7,8-tetrahydroquinazolin-5-amine
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
dimethyl(2-{2-[1-(pyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
3-(1H-imidazol-2-ylmethyl)-6-methoxy-3,4-dihydroquinazolin-4-one
6-[(3-ethoxy-4-methoxyphenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(2S,6S)-4-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-[(3R,4S)-1-(2-aminopyrimidin-4-yl)-4-cyclopropylpyrrolidin-3-yl]-2-cyclopentylacetamide
1-(4-chloro-2-methylphenyl)-5-(2,5-dihydro-1H-pyrrol-2-yl)-3-methyl-1H-1,2,4-triazole