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N-cyclopropyl-2-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyridine-4-carboxamide
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1-(2-methylpropyl)pyrrolidin-2-one
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-phenyl-2-[3-(piperidin-1-yl)pyrrolidin-1-yl]ethane-1,2-dione
1-(2-ethoxyethyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(1H-imidazol-4-yl)ethyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-1-methyl-1H-pyrazole-4-carboxamide
1-{2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(3-chloro-1H-indol-2-yl)methyl]-8-methyl-2,8-diazaspiro[5.5]undecane
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}acetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
N-[(5-chloro-2-methoxyphenyl)methyl]-1-(2-hydroxyethyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
3-chloro-4-fluoro-N-(pyrimidin-4-ylmethyl)-1-benzothiophene-2-carboxamide
ethyl 1-{5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carbonyl}piperidine-4-carboxylate
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
5-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
(3aS,7aR)-5-methyl-2-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-amino-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
ethyl 4-(6,7-dimethoxy-3-{[(thiophen-2-ylmethyl)amino]methyl}quinolin-2-yl)piperazine-1-carboxylate
2-(2-methoxyethyl)-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
N-[2-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)quinolin-6-yl]acetamide
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
2-{5-[(4-chloro-3-methyl-1H-pyrazol-1-yl)methyl]-1-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl}acetamide
1-acetyl-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]piperidine-3-carboxamide
(3R,4R)-N-butyl-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidine-1-carboxamide
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-2,8-dimethylquinoline-4-carboxamide
{4-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]morpholin-2-yl}methanamine
1-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
2-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-6-methylpyridine
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-(1H-pyrazol-1-yl)butanamide
N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-4-methyl-1,4-diazepane-1-carboxamide
4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
4-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidine-4-carbonyl}morpholine
3-(1,3-benzothiazol-2-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]cyclohexanecarboxamide
2-{9-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
5-[1-(1H-imidazol-4-ylmethyl)pyrrolidin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]thiophene-2-carboxamide
1-(4-{4-[(4-methylpentan-2-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
2-[(4-hydroxybutan-2-yl)amino]-N-(propan-2-yl)acetamide
N-(3-ethoxypropyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-(2-chloro-5-sulfamoylphenyl)-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
N-methyl-2-(methylsulfanyl)-N-[1-(pyridin-4-yl)ethyl]-1,3-thiazole-4-carboxamide
N-[3-(6-methoxypyrimidin-4-yl)phenyl]acetamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
(2S,4R)-4-(dimethylamino)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidine-2-carboxylic acid
8-(3-fluorobenzoyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[1-(methoxymethyl)cyclopentyl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
4-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine