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N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]propanamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butan-1-one
3-[(dimethylamino)methyl]-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidin-3-ol
N-({7-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
methyl(oxan-2-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
3-ethyl-1-(2-{[(4-methoxyphenyl)methyl]carbamoyl}ethyl)piperidine-3-carboxylic acid
2-{4-[(4-ethylphenyl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(4-fluorophenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
4-(1-ethyl-1H-pyrazole-3-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
3-(cyclopropylsulfamoyl)-5-[2-(dimethylamino)phenyl]benzoic acid
3-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
2-{[methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-(3-chlorophenyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-ethyl-4,6-dimethyl-3-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
3-[(3R,4S)-4-(dimethylamino)-1-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)piperidin-3-yl]propanoic acid
2-(2-methoxyethyl)-1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
5-[2-(oxolan-3-yl)-1H-imidazol-1-yl]-N-phenylpyridin-2-amine
(4-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(2E)-2-methylbut-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1-{6-[(piperidin-4-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(3S,4R)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
N-ethyl-4-methyl-3-({[(2-propyl-1,3-thiazol-4-yl)methyl]carbamoyl}amino)benzamide
4-[2-(morpholin-4-yl)pyridin-3-yl]-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-({8-[(3-phenoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
3-fluoro-N-({7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
methyl (2R,4S)-4-hydroxy-1-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}piperidine-2-carboxylate
3-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-6-methyl-1,2-dihydroquinolin-2-one
(4aR,8aS)-6-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-{[(5-tert-butyl-2-hydroxyphenyl)methyl](methyl)amino}-N,N-dimethylpropanamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-5-fluoro-1,3-dimethyl-1H-indole-2-carboxamide
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-(3-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
N-[(2S)-1-hydroxypropan-2-yl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
5-{2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
1-[cyclohexyl(methyl)amino]-3-(3-{[(cyclopropylmethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
5-[1-(2H-1,3-benzodioxol-5-yl)-3-(ethoxymethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-1-yl)ethan-1-one
2-{[2-(dimethylsulfamoyl)ethyl]amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
4-methoxy-N-(4-{4-[(pyridin-2-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
1-(3,5-dimethyl-1-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propan-2-yl}-1H-pyrazol-4-yl)ethan-1-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbutanamide
N,5-dimethyl-4-{[(5-methylfuran-2-yl)methyl]amino}-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide