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8-(6-aminohexanoyl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1-[(5-methylfuran-2-yl)methyl]-1,4-dihydropyridin-4-one
8-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-(1-ethyl-1H-pyrazole-5-carbonyl)piperazine
methyl (2R,4S)-4-hydroxy-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine-2-carboxylate
2,3-dimethyl-N-(2-methylquinolin-4-yl)quinoxaline-6-carboxamide
3-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-1-methyl-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}urea
3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
1-[cyclohexyl(methyl)amino]-3-[3-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
1-[(1-{6-[(2,2-dimethylpropyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(1R,2R,4R)-N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
7-[2-(3,4-dichlorophenyl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
4-[(4-fluorophenyl)sulfanyl]-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1-cyclopentyl-3-(3-fluorophenyl)pyrrolidine-2,5-dione
3-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
N,3-dimethyl-4-[({[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}carbamoyl)amino]benzamide
1-{9-[(2,6-dimethylphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl}-2-methoxyethan-1-one
3-(6-chloropyridin-3-yl)-1-[2-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)ethyl]urea
1-cyclopentyl-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,3,4-tetrahydroquinoline-8-carboxamide
2-(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}phenyl)-1H-imidazole
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
2-[3-(4-fluorophenyl)-5-{6-methylpyrazolo[1,5-a]pyrimidin-3-yl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-(3,4-dimethylphenyl)-3-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}urea
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidine-3-carboxylic acid
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-3-phenoxypropan-1-one
3-methyl-1-(4-{1-oxa-8-azaspiro[4.5]decane-8-sulfonyl}phenyl)urea
5-fluoro-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]quinazolin-4-amine
3,4,7-trimethyl-2-(1,4-oxazepane-4-carbonyl)-1H-indole
1-cyclooctyl-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
(2S,4R)-1-(2-methylpropyl)-N-(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(3-{2-[1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(1-ethyl-5-oxopyrrolidin-3-yl)-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
methyl (2S)-1-(4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
{1-[(5-methylthiophen-2-yl)sulfonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(piperidine-1-carbonyl)pyrrolidine-2-carboxylic acid
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-cyclopropylethan-1-one
3-(2-chlorophenyl)-1-(3-methoxypropyl)-3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylfuran-3-carboxamide
1-cyclohexyl-N-(quinolin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
8-(2-chloropyridine-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(2S,3R)-2-amino-1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-hydroxybutan-1-one
3-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}phenol
3-[5-(thiophen-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid