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N-[(3,4-dimethoxyphenyl)methyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,1-benzoxazole
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-2-methylpropanamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
3-{[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]methyl}quinoline
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
6-(2,5-dimethylfuran-3-yl)-N-ethyl-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(4-methylpiperazine-1-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(4-methoxyphenoxymethyl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]propanamide
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[4-(2-methylpropyl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-(2-hydroxyphenyl)-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(3-fluoro-4-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-amino-1-(3,3-diphenylpiperidin-1-yl)-3-hydroxybutan-1-one
1-cyclopentyl-4-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperazin-2-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
(2S)-1-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]pyrrolidine-2-carboxamide
1-[3-(4-fluorophenyl)phenyl]-3-[(5-oxopyrrolidin-2-yl)methyl]-3-(propan-2-yl)urea
4-(benzyloxy)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylbutanamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-butanamido-N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-4-methylbenzamide
3-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propanamide
ethyl 2-{1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-2-yl}acetate
3-(benzylsulfanyl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
2-methyl-5-[3-(1H-pyrazol-3-yl)phenyl]-1,3,4-oxadiazole
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-(2-ethoxyethyl)-3-methyl-5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
4-methyl-2-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidin-3-ol
N-(1-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
N-ethyl-6-(2-methoxyquinolin-3-yl)pyridazin-3-amine
N,N-diethyl-4-(3-methoxy-6-methylpyridin-2-yl)benzene-1-sulfonamide
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-5-{1-[(3E)-hex-3-enoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-(propan-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(3-carbamoyl-4-methoxyphenyl)-1,3-dimethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decane-8-carboxamide
2-(2-chlorophenyl)-N,N-bis(2-hydroxyethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-3-yl)-3-phenylpropan-1-one
2-{1-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}quinolin-4-ol
8-(1-benzofuran-2-ylmethyl)-3-[3-(dimethylamino)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N2-benzyl-6-(2,5-difluorophenyl)-1,3,5-triazine-2,4-diamine
2,6-difluoro-4-methoxy-N-(oxolan-2-ylmethyl)-N-propylbenzamide
(3S,4S)-4-(morpholin-4-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidin-3-ol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(1H-imidazol-1-yl)butan-2-yl]-1H-pyrazole-3-carboxamide
4-(1H-imidazol-1-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]benzamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}pyrrolidine-2-carboxamide
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)propanamide
1-ethyl-3-(morpholine-4-carbonyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one