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1-tert-butyl-4-{[methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
[4-(1-benzyl-1H-pyrazole-4-carbonyl)-1,4-oxazepan-6-yl]methanol
(1S,5R)-6-[6-(methoxymethyl)pyridine-2-carbonyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(naphthalen-1-ylmethyl)-N-(oxolan-2-ylmethyl)-N-propyl-1H-1,2,3-triazole-4-carboxamide
6-{[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]methyl}-1-methyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
[(4aS,8aR)-6-(2,1,3-benzoxadiazol-5-ylmethyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
3-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)propanamide
1-tert-butyl-N-{2-[4-(dimethylamino)phenyl]ethyl}-5-oxopyrrolidine-3-carboxamide
2-(4-{[4-(1H-indole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
N-(1-benzothiophen-2-ylmethyl)-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
4-[(5-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
2-{1-[(2-methylnaphthalen-1-yl)methyl]piperidin-2-yl}acetamide
4-[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]piperazin-2-one
1-ethyl-2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]piperidine
4-[(3,4-difluorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-hydroxyethyl)-3-(3-hydroxyquinoxalin-2-yl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
1-[4-(3-methoxyphenyl)phenyl]-3-(1-methyl-6-oxopiperidin-3-yl)urea
4-[1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]-2-(pyridin-4-yl)pyridine
1-{[1-(naphthalen-2-yl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
1-({1-[6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
(1R,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(cyclohexylsulfanyl)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
2-(2-methoxyethyl)-9-(2-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
1-{2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[2-(5-methylthiophen-2-yl)ethyl]acetamide
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
ethyl[(4-methyl-1H-imidazol-5-yl)methyl][2-(pyrrolidin-1-yl)ethyl]amine
N-({7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
N,6-dimethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-[(2-chloro-6-fluorophenyl)methyl]-N,2-diethyl-4-methyl-1,3-oxazole-5-carboxamide
7-[2-(1,3-benzoxazol-2-ylsulfanyl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4S)-4-amino-1-(2,3-dihydro-1-benzofuran-7-carbonyl)-N-ethylpyrrolidine-2-carboxamide
4-phenyl-3-(piperidin-3-yl)-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methyl-1-benzofuran-7-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
N-[3-({[1-(3-fluoro-4-methoxyphenyl)ethyl]carbamoyl}amino)-2-methylphenyl]-2-methoxyacetamide
2-(1,2-oxazolidin-2-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
N-methyl-N-(oxan-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
(2R,4S)-1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-4-hydroxypiperidine-2-carboxylic acid
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
1-(9H-fluoren-2-ylmethyl)-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-1-methyl-5-oxopyrrolidine-3-carboxamide
5-{imidazo[1,2-a]pyridin-2-yl}-3-[(2-methoxyphenyl)methyl]-1,2,4-oxadiazole
4-{3-[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]propyl}morpholine