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1'-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(pyridin-4-yl)ethyl]acetamide
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
5-methyl-1-(4-methylphenyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
2-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1,4-diazepan-1-yl}-4,6,7-trimethylquinazoline
1-(4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperazin-1-yl)-2-phenoxyethan-1-one
1-{2-[(1-acetylpiperidin-4-yl)oxy]-5-chlorobenzoyl}piperidine-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]propanamide
2-{4-[(1-benzyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyrazine
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenoxy)piperidine
2-(1H-indazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
1-(cyclopentylmethyl)-3-(4-fluorophenyl)pyrrolidine
1-(1-ethyl-1H-pyrazole-3-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{1-[1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]piperidine-3-carbonyl}-4-methylpiperazine
1-[4-(hydroxymethyl)piperidin-1-yl]-2-[4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)morpholin-3-yl]ethan-1-one
N-benzyl-4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonamide
6-(methoxymethyl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)pyridine-2-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,5-dimethylfuran-3-carboxamide
ethyl 4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazine-1-carboxylate
1-{1'-[(2R)-2-amino-2-phenylacetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}piperidin-4-ol
4-{[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
1-benzyl-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-(2,5-dimethylphenyl)-3-[(4,6-dimethylpyrimidin-2-yl)amino]propanamide
1-(furan-2-ylmethyl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]piperidine-4-carboxamide
(3R,4S)-1-(2-methyl-6-propylpyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-amine
3-chloro-6-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyridazine
6-chloro-N,N-dimethyl-3-{[3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
(1R,2S)-2-[(trimethylpyrimidin-4-yl)amino]cyclopentane-1-carboxamide
[(3S,5R)-5-(hydroxymethyl)-1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]piperidin-3-yl]methanol
N-[2-(1H-imidazol-4-yl)ethyl]-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)piperidin-2-one
1,3-dimethyl-6-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-{[(3R,5S)-1-[(3-fluorophenyl)methyl]-5-(morpholine-4-carbonyl)pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
N-[(3-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-chloro-2-methyl-4-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}quinoline
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-cyclopentyl-6-oxopiperidine-3-carboxamide
2-(5-acetylthiophen-3-yl)-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
methyl 4-({[5-(3,4-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}methyl)benzoate
{3-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-oxopropyl}urea
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-phenylazepane-1-carboxamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2,3,6-trimethyl-4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}quinoline
[3-(1H-imidazol-1-yl)propyl][(3-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
7-(1,3-benzothiazol-2-yl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}quinazoline
methyl (2S,4R)-1-[(2-fluorophenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate