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8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[4-methyl-5-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methanol
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(4-fluorophenyl)-2-(piperidin-1-yl)acetamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
4-chloro-3-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
3-(3-fluorophenyl)-3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1-(morpholin-4-yl)-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
7-cyclopropanecarbonyl-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-cyclopentanecarbonyl-N-[2-(pyridin-3-ylformamido)ethyl]piperidine-4-carboxamide
(3S,4S)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-[2-(dimethylamino)ethyl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
ethyl 4-(cyclopropylmethyl)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidine-4-carboxylate
1-benzyl-N3-ethyl-N5-[2-(2-fluorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-({4-methyl-5-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
2-ethoxy-5-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]benzamide
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-(oxolan-3-ylmethyl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
1-(methoxymethyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)cyclobutane-1-carboxamide
{3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-oxopropyl}urea
N-ethyl-5-(1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
[(3-chlorophenyl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-(3-hydroxy-2,2-dimethylpropyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
1-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropane-1-carboxamide
4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2,3,6-trimethylquinoline
4-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(4-chlorophenyl)ethyl]-3-methoxybenzamide
4,6-dimethyl-2-oxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-({[(3R,4R)-1-(2,3-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
2-(2H-1,3-benzodioxol-5-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
N-(3-chlorophenyl)-4-(3-methyl-1,2,4-oxadiazol-5-yl)butanamide
3-(4-chlorophenyl)-N-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N,N-diethyl-1-{[1-(2-methylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(dimethyl-1,3-thiazol-4-yl)-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}acetamide
N-({4-[benzyl(ethyl)amino]quinazolin-2-yl}methyl)-1,2,5-thiadiazole-3-carboxamide
1-methyl-4-(5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-3-phenyl-1H-1,2,4-triazol-1-yl)piperidine
3-{2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[(2-methylphenyl)methyl]-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}acetamide
3-(azocan-1-yl)-N-(2-methylbut-3-yn-2-yl)propanamide
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}quinoxaline-5-carboxamide
2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-ethyl-N-(oxolan-2-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-[2-hydroxy-2-(naphthalen-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-cyclohexyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-pyrazole-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-[(2,5-dimethylphenyl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
N-(2,1,3-benzothiadiazol-5-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-ethoxy-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one