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7-(2-methylphenyl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
(3S,4R)-1-methyl-3-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}piperidin-4-ol
2-(2-methoxyethyl)-9-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
(1S,5R)-6-(morpholine-4-sulfonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
5-{4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
2-benzyl-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
ethyl 1-(cyclohex-3-en-1-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
4-(2-methoxybenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-[3-cyclopentyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
6-cyclopentyl-1-methyl-N-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
5-{[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
1-{1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
1-[5-(ethylsulfanyl)thiophene-2-carbonyl]azepan-3-amine
3-{[(1-benzothiophen-5-ylmethyl)amino]methyl}-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
1-(2-methoxyacetyl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}piperidine-3-carboxamide
4-[4-(4-chlorophenyl)-5-ethyl-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
8-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-hydroxy-3-methylbutanoyl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
4-methyl-6-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1H,2H,3H-pyrazolo[3,4-b]pyridin-3-one
9-(1H-indazole-3-carbonyl)-3-methyl-3,9-diazaspiro[5.6]dodecane
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
N-(4-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}phenyl)acetamide
4-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-oxobutane-1-sulfonamide
1-(3,5-dimethylphenyl)-4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
N-cyclopropyl-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
2-(2,4-dimethoxyphenyl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
methyl 3-(2-ethylbutanoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-benzyl-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1,3-benzoxazole-5-carboxamide
N-(2-methoxyethyl)-1-methyl-N-(pyridin-3-ylmethyl)azepane-2-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[5-(2,4-difluorophenoxymethyl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
(2E)-1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-ethyl-1-[(2-fluorophenyl)methyl]-6-oxo-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
3-hydroxy-3-phenyl-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
(3S,5S)-1-(3-methylbenzoyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
8-[(3-methoxyphenyl)methyl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aR,6aR)-2-[2-(2-chloro-4-fluorophenyl)acetyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(1,2-oxazinan-2-yl)propanamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide