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1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
2-{2-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenoxy}propanoic acid
N-butyl-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(hydroxymethyl)azepan-4-ol
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(2-phenoxyethyl)piperazine
3-{2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-4-[(4-methylphenyl)methyl]piperazin-2-one
3-(3-{3-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)propan-1-ol
4-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}benzoic acid
ethyl 1-(7-chloroquinolin-4-yl)-5-{[(oxolan-2-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
{1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
3-hydroxy-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
6-(2-aminoethyl)-2-{4-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-ylmethyl]phenyl}-3,4-dihydropyrimidin-4-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-[2-(methylsulfanyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[(4-ethoxyphenyl)methyl]-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
4-benzoyl-1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
3-methyl-1-(3-methylcinnolin-5-yl)-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
1-butyl-3-cyclopentyl-5-(1,4-dioxan-2-yl)-1H-1,2,4-triazole
4-benzyl-1-(5-chloro-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-ethyl-1,4-diazepan-5-one
2-[(2R)-2-aminopropanoyl]-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(1-methoxybutan-2-yl)benzamide
5-(3-methylthiophene-2-carbonyl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{5-[(1S)-1-amino-2-cyclohexylethyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl}benzamide
(3S,4S)-4-(morpholin-4-yl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrrolidin-3-ol
3-(oxolan-3-yl)-5-{pyrazolo[1,5-a]pyridin-3-yl}-1,2,4-oxadiazole
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
1-[(4,6-dimethylquinolin-2-yl)amino]-3-ethoxypropan-2-ol
4-(methoxymethyl)-6-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
5-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
3-{5-[(dimethyl-1,2-oxazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(2-hydroxyethyl)propanamide
2-{methyl[2-(pyridin-2-yl)ethyl]amino}-2-(4-methylphenyl)acetic acid
5-(2-chloro-4-methoxyphenoxymethyl)-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-ethyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
4-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
1-cyclobutanecarbonyl-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[5-(hydroxymethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
6-(2-methoxyphenyl)-3,4-dihydroquinazolin-4-one
N-(carbamoylmethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-(4-fluorophenoxymethyl)pyrimidin-4-ol
methyl 6-[(3,5-dimethylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S)-3-(1H-imidazol-4-yl)-2-{[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]formamido}propanamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
2-(azepane-1-carbonyl)-6-(3-chlorophenyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-{1-[(2Z)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decane
[4-(4-methyl-5-phenylthiophene-2-carbonyl)-1,4-oxazepan-6-yl]methanol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,3-thiazole-5-carboxamide