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1-(3-{[ethyl(2-hydroxyethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]benzamide
5-[1-(dimethyl-1H-1,2,4-triazol-1-yl)propan-2-yl]-1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazole
1-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-1,2,3-triazole
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
N-[2-(ethylsulfanyl)ethyl]-4-{[(2R)-2-hydroxypropyl]sulfamoyl}benzamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}propanamide
4-benzyl-1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1,4-diazepan-5-one
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(3-methylpyridin-4-yl)methyl]benzamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-ethyl-5-{methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(2,3,6-trifluorophenyl)methyl]amine
2-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}formamido)-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
4-(1H-imidazole-2-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
methyl[(4-phenoxyphenyl)methyl]{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(3R,4S)-4-phenyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-amine
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
4,4,4-trifluoro-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{4-[({[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]phenyl}pyrrolidin-2-one
[(3S,5R)-1-(dimethyl-1,2-oxazole-4-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
N-methyl-N-[1-(pyridin-4-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-[2-(4-fluorophenyl)morpholin-4-yl]-4-oxobutane-1-sulfonamide
methyl 3-[(3S,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
[(3R,4S)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)({[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl})methylamine
N-ethyl-N-[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-(phenylsulfanyl)acetamide
1-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidin-3-ol
4-(2-fluoro-3-methoxyphenyl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
{9-[(5-methylthiophen-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
2-(2-aminoethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]quinazolin-4-amine
N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-ethyl-8-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(pyridin-4-yl)propanamide
1-(4-{[2-(ethylsulfanyl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]cyclopent-1-ene-1-carboxamide
9-{6-methylthieno[2,3-d]pyrimidin-4-yl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
7-methyl-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidin-2-amine
methyl 4-{3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamido}butanoate
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(1R,5R)-6-(3-phenoxypropyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-[5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]butan-1-amine
1-(4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}thiophen-2-yl)ethan-1-one