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ethyl 6-({4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate
4-benzyl-3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-chloro-N-methyl-6-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,6-dihydropyridine-3-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[4-(quinoxalin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
2-[5-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl]acetic acid
methyl 1-methoxy-2-oxo-8-[(4-oxo-4H-chromen-3-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
(3S,9aR)-8-[(5-chlorothiophen-2-yl)methyl]-3-(cyclohexylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(3,5-difluorobenzoyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-chloro-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
4-[(4-fluorophenyl)methyl]-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine
3-(2-methylphenoxy)-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
N-[1-(7-{[4-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-methoxybenzamide
1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-(4-methylphenoxymethyl)piperidine
2-amino-6-(propan-2-yl)-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}pyridine-3-carbonitrile
2-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-benzyl-N-[2-(dimethylamino)ethyl]-2-(1-methylpiperidin-2-yl)acetamide
N-(1-hydroxy-2-methylpropan-2-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(1S,5R)-3-(1H-imidazol-4-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrido[2,3-d]pyrimidin-4-amine
N-cyclopropyl-4-methoxy-3-[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
1-cyclobutanecarbonyl-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]piperidine-4-carboxamide
1-(3-chloro-4-methoxyphenyl)-2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-(4-methoxy-2-methylphenyl)-3-{1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl}propanamide
8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-fluorophenyl)piperazine
3-(2-ethyl-1H-imidazol-1-yl)-N-(3-phenylprop-2-yn-1-yl)-N-propylpropanamide
4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-3-(3-methylphenyl)-1H-pyrazole
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(3,3-diphenylpropyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(azepane-1-carbonyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzene-1-sulfonamide
2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)acetamide
(1S,5R)-3-(4-methoxybenzenesulfonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
1-[(2-fluorophenyl)methyl]-N-[(3-methyloxetan-3-yl)methyl]-6-oxopiperidine-3-carboxamide
(1S,5R)-3-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}acetamide
1,4,6-trimethyl-3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
3-{[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole-4-sulfonamide
2-[3-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
3-chloro-N-(4-{4-[(1-methoxypropan-2-yl)amino]piperidin-1-yl}phenyl)benzamide
7-(5-chloro-2-methoxyphenyl)-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-7-methyl-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}quinoline
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}spiro[2.2]pentane-1-carboxamide