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N-[(4-chlorophenyl)(phenyl)methyl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)acetamide
2-methyl-5-[4-(quinoline-8-sulfonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-(2-fluorophenyl)-1H-pyrazole
4-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-2-(trifluoromethyl)morpholine
benzyl(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-(1-methyl-2-oxopyrrolidin-3-yl)-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carboxamide
5-(3-fluorophenoxymethyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
(3S,9aR)-8-benzoyl-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]pyridine-3-carbonitrile
[(3R,4R)-1-(pyridine-3-sulfonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-(3-{[(cyclobutylmethyl)(oxolan-2-ylmethyl)amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
(1R,7S)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[(3aS,6aS)-2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-methyl-2-(1-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)-N-[3-(oxolan-2-yl)propyl]acetamide
(4aR,7aS)-1-ethyl-4-(3-methoxy-5-methylthiophene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(1S,2R)-2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]-1-hydroxypropyl]phenol
{4-[(4-methoxyphenyl)methyl]-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl}methanol
4-[1-(2-phenylethyl)pyrrolidin-3-yl]-N-(prop-2-en-1-yl)piperidine-1-carboxamide
2-{3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]piperidin-1-yl}acetamide
4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyridine-4-carbonyl}morpholine
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
({5-[1-(4-fluoro-3-methylbenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(2-methyl-1,3-benzothiazol-6-yl)-2,3-dihydro-1H-isoindole-1,3-dione
(5S)-1,2,2,5-tetramethyl-4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazine
2-methyl-4-(5-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
1-(2-oxo-2-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
2-cyclopropyl-9-(1,2-oxazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
2-(1,2,3,4-tetrahydroisoquinolin-2-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}propanamide
3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
4-(2,3-difluorobenzoyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrazine-2-carboxamide
N-methyl-N-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)oxolan-3-amine
(4aS,7aR)-1-(2-ethylpyrimidine-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 1-benzyl-3-(oxolane-2-amido)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[2-(4-fluorophenyl)ethyl]-4-[4-(naphthalene-1-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-3-(1H-pyrazol-5-yl)piperidine
3-(4-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}piperazin-1-yl)propan-1-ol
{1-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
3-{[4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazin-1-yl]methyl}benzoic acid
{2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}urea
(1R,5S)-3-(5-propyl-1,2-oxazole-3-carbonyl)-3,8-diazabicyclo[3.2.1]octane
3-(6-amino-2-methylpyridin-3-yl)phenol
3-(4-{[4-(2-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)benzonitrile
N-cyclopropyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}quinoline-8-sulfonamide
3-(3-fluorophenyl)-1-methyl-3-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
(3R,4R)-1-(benzenesulfonyl)-4-{[2-(3-methylpyridin-2-yl)ethyl]amino}pyrrolidin-3-ol
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrimidin-4-amine
2-(furan-3-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-imidazole