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1-({[3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclohexanecarboxamide
{1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-(1H-indol-4-ylmethyl)-1-benzofuran-2-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-cyclopentyl-N-methyl-6-oxopiperidine-3-carboxamide
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-4-yl)pyridine
3-(2-fluorophenyl)-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-phenylpropanamide
N-{4-[2-(dimethylamino)ethoxy]-1-(4-fluorophenyl)-1H-indazol-3-yl}-1H-pyrazole-3-carboxamide
1-(2,4-dimethylphenoxy)-3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)propan-2-ol
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(2-phenylethyl)piperidine
N-methyl-N-(2-methylpropyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
7-methyl-2-(5-phenoxyfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3R,4S)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-amine
(1R,2S)-N-methyl-2-[4-(4-methylphenoxy)piperidine-1-carbonyl]cyclohexane-1-carboxamide
8-[(4-methoxy-3-methylphenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(2S)-2-amino-1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-hydroxypropan-1-one
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-3-yl]-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
(1R,3S)-7-(3-ethoxybenzoyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-ethoxy-3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]pyridine
N-ethyl-N-(pyridin-4-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
(4aR,7aS)-4-[2-(furan-2-yl)-2-oxoacetyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2R,3S,6R)-5-benzoyl-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4,6-dimethylpyrimidin-2-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]piperidin-4-amine
(3aS,7aR)-2-(8-fluoro-4-oxo-1,4-dihydroquinoline-3-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(1-propylpiperidin-4-yl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
(2R,3R,6R)-3-(3,5-difluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
3-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoic acid
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-2,1,3-benzothiadiazole-4-sulfonamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
2-(3-methoxypropyl)-9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
8-(1H-indol-5-ylmethyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(4-chlorophenyl)methyl]-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{[1-(dimethylamino)cyclohexyl]methyl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
methyl (2S)-2-[(7-fluoro-3-methyl-1-benzofuran-2-yl)formamido]-4-methylpentanoate
(2S,4S)-4-amino-N-[(4-methoxynaphthalen-1-yl)methyl]-N,1-dimethylpyrrolidine-2-carboxamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(8-methyl-2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}quinolin-3-yl)methanol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
3-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-5-phenyl-1,2,4-oxadiazole
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
(1S,6R)-9-(2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
3-propyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
2,8-dimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]quinoline-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
8-(1-benzoxepine-4-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine