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N-(propan-2-yl)-6-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazin-1-yl)pyrimidin-4-amine
4-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(4-methylphenyl)-1H-pyrazole
N-(1,3-benzothiazol-5-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
N-(3-methoxypropyl)-1-methyl-N-(1,3-thiazol-4-ylmethyl)piperidin-4-amine
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-fluoro-3-methyl-1H-indole
2-(2-chloro-4-fluorophenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
2-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
9-(cyclopropylmethyl)-1-methyl-4-(9H-purin-6-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(2-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)sulfanyl]pyridine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-{2-[(propan-2-yl)carbamoyl]ethyl}pyrrolidin-3-yl]-1-methyl-1H-imidazole-2-carboxamide
(1S,5R)-3-(2,6-difluoro-4-methoxybenzoyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
1-benzyl-5-acetamido-N,2-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
N-(6-methylpyridin-3-yl)-3-(thiophen-3-yl)propanamide
5-methoxy-3-methyl-2-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-1H-indole
2-(3-{[(butan-2-yl)(cyclopentyl)amino]methyl}phenoxy)acetamide
4-methyl-3-{pyrazolo[1,5-a]pyridin-7-yl}-1,2-dihydroquinolin-2-one
3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propanoic acid
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1-cyclopentyl-3-(3-fluorophenyl)pyrrolidine-2,5-dione
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
(4aR,7aS)-1-benzyl-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-4-{4-[3-(pyridin-3-yloxy)azetidine-1-carbonyl]phenyl}butan-2-ol
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
5-[4-(4-ethylpiperazin-1-yl)piperidine-1-carbonyl]-1-[(2-fluorophenyl)methyl]piperidin-2-one
ethyl 4-(2-methoxyethyl)-1-[1-(2-methoxyphenyl)propan-2-yl]piperidine-4-carboxylate
3,7-dimethyl-11-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-3,7,11-triazaspiro[5.6]dodecane
2-(piperidin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethan-1-one
1-[4-(4-{[2-(1H-imidazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]-3-methylimidazolidin-2-one
4-(4-{bicyclo[2.2.1]hept-5-en-2-ylmethyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
9-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
[4-(4-methoxyphenyl)butan-2-yl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
4-(5-methyl-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)piperazine-1-carbaldehyde
2-(pyridin-3-ylmethyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(4-chlorophenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-{1-[(2,4,5-trimethoxyphenyl)methyl]pyrrolidin-2-yl}ethan-1-ol
2-(3-methanesulfonylpropanoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
(3S,4S)-1-[3-(2-oxopyrrolidin-1-yl)benzoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-benzyl-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{4-[2-(2-phenylethyl)morpholin-4-yl]piperidin-1-yl}ethan-1-one
2-amino-4-[2-(2-methylphenyl)pyrimidin-5-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
3-(3-hydroxy-3-methylbutyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
3-(4-acetamidophenyl)-4-methoxybenzamide