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N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
N-benzyl-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-ethylbenzamide
3-[(5-ethylfuran-2-yl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(1-ethylpiperidin-4-yl)-2,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
1-[(4-methoxy-3-methylphenyl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-(3-chloro-4-fluorophenoxy)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methyl-1,3-benzothiazol-6-yl)pyrrolidine-1-carboxamide
(2R,6S)-2,6-dimethyl-4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}morpholine
1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
1-(4-chloro-1H-pyrrole-2-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
(4aS,8aS)-2-(6-aminopyrimidin-4-yl)-7-(propane-1-sulfonyl)-decahydro-2,7-naphthyridin-4a-ol
7-methoxy-3-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(4-{[4-(thian-4-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-{[3-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)-N-(prop-2-en-1-yl)benzamide
N-cyclobutyl-3-{[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]sulfamoyl}benzamide
3-[2-(dimethylamino)ethyl]-8-[3-(morpholin-4-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3,5-dichloro-4-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyridine
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]acetamide
4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]benzene-1-sulfonamide
2-ethyl-5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-4-methyl-1,3-oxazole
3-(1,2-oxazinan-2-yl)-1-[3-(3-phenylpropanoyl)piperidin-1-yl]propan-1-one
(3S,4R)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-({7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
2-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
diethyl[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
methyl 3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]propanoate
2,6-dimethyl-5-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-[3-(4-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-ol
5-[1-(1H-pyrazol-1-yl)ethyl]-3-(thiophen-2-yl)-1,2,4-oxadiazole
2-butyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
(3S,9aR)-8-(3-chlorobenzoyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,5-dimethyl-3-(3-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
N-[5-({[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)-2-methylphenyl]-2-(dimethylamino)acetamide
3-[2-(N-methylmethanesulfonamido)ethyl]-1-[2-(methylsulfanyl)phenyl]urea
3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[(3-methylthiophen-2-yl)methyl]piperidine-3-carboxylic acid
N-methyl-5-({4-[1-(N-methylacetamido)ethyl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
4-(4-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
5-ethyl-2-[1-(6-methoxypyridin-3-yl)-1H-imidazol-2-yl]pyridine
1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonitrile
4-(2-chloro-4-fluorobenzoyl)-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-fluoro-4-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-(trifluoromethyl)pyrimidin-4-amine