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N-methyl-5-[(methylsulfanyl)methyl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}furan-2-carboxamide
2-(1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
2-hydroxy-N-{2-[4-(1H-imidazol-4-ylmethyl)morpholin-2-yl]ethyl}benzamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)-1H-imidazole
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(oxolan-2-ylmethyl)pyridin-2-amine
1-(3,5-dimethylphenyl)-4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
1'-[(2-methyl-1,3-oxazol-4-yl)methyl]spiro[indene-1,4'-piperidine]
2-(dimethyl-1,3-thiazol-5-yl)-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)acetamide
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-5-methoxy-3,4-dihydroquinazolin-4-one
2-methyl-8-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(2,3-dimethylquinoxalin-6-yl)formamido]acetic acid
2-[(2-amino-6-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-yl)amino]ethan-1-ol
N-methyl-N-({1-[(2,4,5-trifluorophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
1-cyclohexyl-1-[2-(ethylsulfanyl)ethyl]-3-(3-sulfamoylphenyl)urea
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-6-(piperidin-1-yl)pyrimidin-4-amine
N-cyclopropyl-1-{1-[2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}piperidine-3-carboxamide
2-[({5-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
1-methyl-4-{1-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]ethyl}piperazine
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methoxybenzoyl)piperazine
(2S,4R)-4-amino-1-(1,4-dimethylpiperidine-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-[2-(2-ethylphenyl)pyridin-3-yl]cyclopropanecarboxamide
1-phenyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-1,2,3-triazole-5-carboxamide
N,N-diethyl-2-{4-[(2S)-4-ethyl-2-methyl-3-oxopiperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
(3S)-N,N-dimethyl-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]azepan-3-amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
6-oxo-N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]piperidine-3-carboxamide
N-(3,3-diphenylpropyl)-6-[(2-hydroxy-4-methoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[(4aR,8aS)-1-(2,7,8-trimethylquinoline-4-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
3-{[2-(2-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-4H-chromen-4-one
2-ethyl-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(4,5-dichloro-1H-imidazol-1-yl)acetamide
1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
methyl 5-{[(4-acetamidophenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(2-methylphenyl)-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one
5-[(3-methoxyphenyl)methyl]-3-methyl-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-[(3-chlorophenyl)methyl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
(1S,5R)-3-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(3,4-difluorophenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N,1-dimethyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]ethyl}-1H-pyrazole-3-carboxamide
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-5-phenyl-1,2-oxazole
N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)oxan-4-amine
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(1-methyl-1H-pyrazol-5-yl)propanamide
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
1-{2-[(6-methoxypyrimidin-4-yl)oxy]hex-5-en-1-yl}-4-methyl-1,4-diazepane
methyl 1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-{[5-(4-hydroxyphenyl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
3-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
(3S,4S)-1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol