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N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
5-(2-methyl-1,3-thiazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-cyclobutyl-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
2-(dimethylamino)-4-methyl-N-[1-(pyridin-4-yl)propyl]pyrimidine-5-carboxamide
2-{5-cyclopropyl-4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(5-methylfuran-2-yl)pyrimidine
N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]-1,4-dioxane-2-carboxamide
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
3-{[4-(dimethylamino)-5-methylpyrimidin-2-yl](methyl)amino}propane-1,2-diol
[5-({7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)furan-2-yl]methanol
1-(4-methylpiperidin-1-yl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylpyridine
[(3R,4R)-1-[3-(difluoromethoxy)benzoyl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-(cyclohexylmethyl)-5-(cyclopentylamino)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[7-fluoro-2-(thiophen-3-yl)quinolin-3-yl]methyl}[2-(3-methoxyphenyl)ethyl]amine
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-cyclopropylpyrimidine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-methylacetamide
{1-[3-(5-fluoropyrimidin-2-yl)phenyl]ethyl}dimethylamine
3-[5-(2,4-dimethoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-(3-chloro-4-methoxyphenyl)-6-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
N-methyl-N-(pyridin-3-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
(4aS,7aR)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 3-acetamido-1-ethyl-5-{[(4-fluorophenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
5-(dimethylamino)-2-[2-(naphthalen-2-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
2-acetyl-8-[(2,3-difluoro-4-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3-hydroxyphenyl)methyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(3,4-dimethylphenyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-hydroxy-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propan-1-one
methyl 3-[(3S,4R)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoate
5-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
(2S)-2-hydroxy-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(2-methylpropyl)(oxolan-2-ylmethyl)amine
4-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)carbamoyl)amino]-N,3-dimethylbenzamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-chloropyridine-4-carboxamide
2-chloro-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}pyridin-3-amine
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}ethan-1-one
4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
2-[1-(3-methylbut-2-en-1-yl)-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(propylsulfanyl)ethan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(3-hydroxy-3-methylbutyl)benzamide
2-[4-({[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
2-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
5-methyl-N-(2-methylpropyl)-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-cyclopropyl-N-(furan-3-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine