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N-(4-methylpentan-2-yl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
methyl 5-[(2,3-difluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
2-(3-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}phenoxy)acetamide
ethyl 4-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine-1-carboxylate
1-(2,2-dimethylpropyl)-4-[(1H-imidazol-2-ylmethyl)amino]pyrrolidin-2-one
5-[3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-oxopropyl]-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
2-ethyl-9-(2-methylpyrimidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
9-methoxy-7-[4-(methylsulfanyl)phenyl]-4-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(1R,2R,4R)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-ethenyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]benzamide
2,4-dimethyl-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
methyl 1-({4-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperidine-4-carboxylate
N-[1-(furan-2-carbonyl)piperidin-3-yl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{2-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
1-(4-chloro-3-methylbenzoyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
diethyl({[3-(2-phenylazetidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(4-fluorophenyl)-1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]ethyl]methylamine
1-{[(3R,4R)-1-(2-chloro-4-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
5-(furan-2-yl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
1-[4-({4-[3-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[4-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-[(4-chlorophenyl)methyl]-5-(pyrrolidine-1-carbonyl)-1,3-benzoxazole
(5S,9aS,9bS)-2-(2-phenylethyl)-5-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
9-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-6-oxa-9-azaspiro[4.5]decane
3-({[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-1-(2-methoxyphenyl)piperazin-2-one
8-[(6-chloropyridin-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[2-(benzylamino)ethyl]-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)-N,N,6-trimethylpyrimidin-2-amine
N-[4-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]acetamide
4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(2R,3R)-1'-(dimethyl-1,3-thiazole-5-carbonyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
5-cyclobutyl-N-[2-(3-methylthiophen-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
[(1-benzylpyrrolidin-3-yl)methyl][(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
2-{2-methyl-3-[({2-[(3-methylpyridin-2-yl)amino]ethyl}amino)methyl]-1H-indol-1-yl}acetamide
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(2-phenylindolizin-3-yl)ethane-1,2-dione
2,4-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,3-thiazole-5-carboxamide
5-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
2-hydroxy-2-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]propanamide
(3aS,6aS)-2-[(4-fluorophenyl)methanesulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid