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4-[(2-butoxy-3-methoxyphenyl)methyl]-3-methylpiperazin-2-one
6-(3-methoxyphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-({1-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azonane
N-[2-(dimethylamino)ethyl]-3-({1-[(4-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-4-methylpiperazine-1-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
4-(4-methoxyphenyl)-2-methyl-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazine
N-{[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenylacetamide
(5S)-5-(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidine-1-carbonyl)pyrrolidin-2-one
3-[(3,4-difluorophenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
2-phenoxy-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}acetamide
methyl 2-[(4-fluorophenyl)sulfamoyl]-6-(2-methylbutyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{[(2E)-2-methylbut-2-en-1-yl](thiophen-2-ylmethyl)amino}ethan-1-ol
5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-2-(pyridin-3-yl)acetamide
2-cyclopropyl-N-[1-(2-fluorophenyl)piperidin-4-yl]-1,3-benzoxazole-6-carboxamide
1-(2-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}ethyl)pyrrolidin-2-one
2-amino-N-(isoquinolin-5-ylmethyl)-N,4-dimethyl-1,3-benzothiazole-6-carboxamide
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
methyl(pyrazin-2-ylmethyl){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
N-cyclopropyl-3-{[3-(pyridin-3-yl)propyl]sulfamoyl}benzamide
(4aS,7aR)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-methanesulfonylethyl)-5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazole
2-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl}benzoic acid
2-(2,5-dimethylphenyl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(4-ethyl-1H-pyrazol-5-yl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[2-(3-fluorophenyl)ethyl]-1-[(4-fluorophenyl)methyl]pyrrolidine-2-carboxamide
3-phenyl-4-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1H-pyrazole
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
ethyl 4-benzyl-1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidine-4-carboxylate
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-2-one
1-[4-(difluoromethoxy)benzoyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
9-methoxy-4-(4-methoxybenzenesulfonyl)-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,4R)-1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-methyl-4-(1-phenyl-1H-pyrazol-5-yl)-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-oxo-1-(2-phenylethyl)-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
1-[4-(azepan-1-yl)-4-oxobutanoyl]-3-ethylpiperidine-3-carboxylic acid
(1S,5R)-3-{2-[cyclopentyl(methyl)amino]acetyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(furan-2-ylmethyl)-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-4-carboxamide
2-{[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}-N-methylbutanamide
methyl 3-({[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)propanoate
4-[(5-{[3-(benzyloxy)propyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}benzoic acid
(3S,4S)-1-(9H-fluoren-2-ylmethyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
1-cyclopentyl-5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-N-methyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
N-methyl-2-(1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3-oxopiperazin-2-yl)acetamide